Pyrazole

Pyrazole

SCHEMBL360175

COc1ccc2ncsc2c1.c1cn[nH]c1

nearest known ligand 0.49

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 6/20 0.49
RAB9A P51151 6/20 0.49
ALDH1A1 P00352 6/20 0.49
MEN1 O00255 5/20 0.49
KMT2A Q03164 5/20 0.49
SMN1; SMN2 Q16637 5/20 0.49
KDM4E B2RXH2 3/20 0.49
HPGD P15428 1/20 0.49
TDP1 Q9NUW8 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.41
MAPT P10636 6/20 0.39
NFKB1 P19838 1/20 0.39
NFKB2 Q00653 1/20 0.39
RELA Q04206 1/20 0.39
HTT P42858 2/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C19 P33261 1/20 0.39
LMNA P02545 1/20 0.39
PFKFB3 Q16875 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23133 0.85 NPC1 (0.57) NPC1RAB9AALDH1A1MEN1KMT2A
Bromide SCHEMBL1193036 0.83 NPC1 (0.56) NPC1RAB9AALDH1A1MEN1KMT2A
Toluene SCHEMBL11239856 0.78 ALDH1A1 (0.49) NPC1RAB9AALDH1A1MEN1KMT2A
Benzo[D]Thiazole SCHEMBL360258 0.77 ALDH1A1 (0.66) NPC1RAB9AALDH1A1SMN1; SMN2KDM4E
SCHEMBL29992983 0.73 NPC1 (0.56) NPC1RAB9AALDH1A1MEN1KMT2A
SCHEMBL11719234 0.73 RIPK2 (0.47) NPC1RAB9AALDH1A1MEN1KMT2A
SCHEMBL29967146 0.72 NPC1 (0.47) NPC1RAB9AALDH1A1MEN1KMT2A
SCHEMBL928266 0.72 NPC1 (0.47) NPC1RAB9AALDH1A1MEN1KMT2A
SCHEMBL8433660 0.71 MEN1 (0.46) NPC1RAB9AALDH1A1MEN1KMT2A
SCHEMBL6032519 0.70 RAB9A (0.46) NPC1RAB9AALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012007510-A1 COMPOUNDS FOR BINDING AND IMAGING AMYLOID PLAQUES AND THEIR USE BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2012-01-19 WO disclosed