SCHEMBL3603674

SCHEMBL3603674

COC(=O)c1cc2ccc(-c3ccc(C)cc3)cc2n1CC(=O)NCCNCC1CCCCC1

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 3/20 0.41
MTNR1B P49286 3/20 0.41
NPC1 O15118 2/20 0.39
AVPR1B P47901 2/20 0.39
RAB9A P51151 1/20 0.39
CNR1 P21554 1/20 0.38
MMP13 P45452 1/20 0.37
GSK3B P49841 1/20 0.37
NPSR1 Q6W5P4 2/20 0.36
TP53 P04637 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
GAA P10253 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
TSHR P16473 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3609348 0.91 NPC1 (0.40) NPC1AVPR1BRAB9ACNR1MMP13
SCHEMBL3603676 0.84 MTNR1A (0.40) MTNR1AMTNR1BNPSR1TP53GAA
SCHEMBL3602467 0.81 KDM4E (0.46) NPC1RAB9ACNR1MMP13NPSR1
SCHEMBL3591928 0.79 GRIN2B (0.46) NPC1RAB9ACNR1NPSR1SMN1; SMN2
SCHEMBL3586999 0.79 KMT2A (0.49) NPC1RAB9A
SCHEMBL3586855 0.79 BRD4 (0.44) NPC1RAB9ACNR1SMN1; SMN2L3MBTL1
SCHEMBL3596258 0.79 NPC1 (0.47) NPC1RAB9ACNR1
SCHEMBL13115992 0.76 HPGD (0.38) GSK3BNPSR1TP53SMN1; SMN2GAA
SCHEMBL3599501 0.75 GPR35 (0.38) GSK3BNPSR1TP53SMN1; SMN2GAA
SCHEMBL3644326 0.75 KDM4E (0.48) MTNR1AMTNR1BNPSR1SMN1; SMN2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7807704-B2 Bicyclic, nitrogen-containing compounds modulating CXCR4 and/or CCXCKR2 CHEMOCENTRYX, INC. (US) 2010-10-05 US disclosed
US-20070275965-A1 CXCR4 modulators CHEMOCENTRYX, INC. (US) 2007-11-29 US disclosed
WO-2007115231-A2 CXCR4 MODULATORS CHEMOCENTRYX, INC. (US) 2007-10-11 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070275965-A1 CXCR4 modulators CXCL12, CXCR4, CXCR1 MTNR1A 1079/4885MTNR1B 833/4885NPC1 334/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.