SCHEMBL3605880

SCHEMBL3605880

C[C@H](N)c1c(-c2ccc(Cl)cc2Cl)ncn1CCc1c[nH]c2ccccc12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MDM4 O15151 2/20 0.43
MDM2 Q00987 2/20 0.43
HDAC8 Q9BY41 1/20 0.43
TP53 P04637 1/20 0.43
NR3C1 P04150 4/20 0.41
NR3C2 P08235 3/20 0.41
PGR P06401 1/20 0.41
GOT1 P17174 1/20 0.40
HTR2A P28223 2/20 0.40
ADRB1 P08588 1/20 0.40
HTR1A P08908 1/20 0.40
ADRA2A P08913 1/20 0.40
SLC6A2 P23975 1/20 0.40
HTR1D P28221 1/20 0.40
HTR1B P28222 1/20 0.40
HTR2C P28335 1/20 0.40
HTR1E P28566 1/20 0.40
SLC6A4 P31645 1/20 0.40
HTR7 P34969 1/20 0.40
HTR2B P41595 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3607898 0.92 MDM2 (0.46) MDM4MDM2HDAC8TP53HTR2A
SCHEMBL3598443 0.88 HTR2A (0.42) MDM4MDM2TP53HTR2AHTR1A
SCHEMBL3604686 0.85 DPP4 (0.41) HDAC8TP53GOT1HTR2AHTR1D
SCHEMBL3599723 0.84 CNR1 (0.42) MDM4MDM2TP53SLC6A2SLC6A4
SCHEMBL3594733 0.81 CXCR2 (0.44) MDM4MDM2TP53NPC1GAA
SCHEMBL3595829 0.78 CYP3A4 (0.44) MDM4MDM2TP53RAB9A
SCHEMBL3595338 0.78 PNMT (0.41) HTR6MAPT
SCHEMBL3597273 0.77 CXCR2 (0.40) MDM4MDM2HDAC8TP53MEN1
SCHEMBL3599359 0.76 CXCR2 (0.40) MDM4MDM2HDAC8TP53MEN1
SCHEMBL3600935 0.76 TP53 (0.45) MDM4MDM2TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7728146-B2 Enzyme inhibitors PROBIODRUG AG (DE) 2010-06-01 US claimed