SCHEMBL3605672

SCHEMBL3605672

CC(C)(C)OC(=O)N1CCc2cc(C(=O)Nc3cnn(Cc4cccc5ccccc45)c3)ccc2C1

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SCD O00767 2/20 0.48
SCD5 Q86SK9 1/20 0.48
NAMPT P43490 6/20 0.45
ESR2 Q92731 1/20 0.44
TMPRSS2 O15393 2/20 0.42
ACHE P22303 1/20 0.42
RPS6KA2 Q15349 1/20 0.42
ALDH1A1 P00352 1/20 0.41
KDM4E B2RXH2 1/20 0.40
USP2 O75604 1/20 0.40
HPGD P15428 1/20 0.40
MAPK1 P28482 1/20 0.40
JAK2 O60674 1/20 0.40
JAK3 P52333 1/20 0.40
PTK2 Q05397 1/20 0.40
NR1H2 P55055 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3596141 0.92 TMPRSS2 (0.47) SCDSCD5NAMPTESR2TMPRSS2
SCHEMBL3606130 0.90 KDM4E (0.50) SCDSCD5NAMPTESR2RPS6KA2
SCHEMBL3601224 0.89 SCD5 (0.51) SCDSCD5NAMPTESR2ALDH1A1
SCHEMBL3615748 0.84 SCD (0.53) SCDSCD5NAMPTESR2RPS6KA2
SCHEMBL3602942 0.84 MEN1 (0.51) SCDSCD5NAMPTESR2TMPRSS2
SCHEMBL3605783 0.84 NAMPT (0.56) SCDSCD5NAMPT
SCHEMBL3605404 0.84 NAMPT (0.63) SCDSCD5NAMPTESR2ALDH1A1
SCHEMBL3599020 0.83 SMN1; SMN2 (0.57) SCDSCD5NAMPTESR2TMPRSS2
SCHEMBL3603596 0.83 SCD (0.53) SCDSCD5NAMPTESR2TMPRSS2
SCHEMBL3602755 0.83 SCD (0.51) SCDSCD5NAMPTESR2TMPRSS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100041696-A1 Compounds SMITHKLINE BEECHAM CORPORATION 2010-02-18 US disclosed
US-20100041696-A1 Compounds SMITHKLINE BEECHAM CORPORATION 2010-02-18 US disclosed
US-20100041696-A1 Compounds SMITHKLINE BEECHAM CORPORATION 2010-02-18 US disclosed
WO-2008074824-A2 ISOQUINOLINECARBOXAMIDES AS INHIBITORS OF STEAROYL-COA DESATURASE (SCD) SMITHKLINE BEECHAM CORPORATION (US) 2008-06-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100041696-A1 Compounds CYP11B2, SCD, CYP3A5 SCD 2/4885SCD5 4/4885NAMPT 869/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.