SCHEMBL360587

SCHEMBL360587

O=Cc1ccc(N2CCC3(CCC(CC(=O)O)CC3)CC2)nc1

nearest known ligand 0.57

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
FFAR4 Q5NUL3 18/20 0.57
DGAT1 O75907 2/20 0.54
CYP3A4 P08684 1/20 0.54
CYP2C9 P11712 1/20 0.54
KCNH2 Q12809 1/20 0.54
FFAR1 O14842 1/20 0.53
ACAT1 P24752 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19134108 0.81 FFAR4 (0.65) FFAR4CYP3A4CYP2C9FFAR1
SCHEMBL14127679 0.80 DGAT1 (0.61) DGAT1KCNH2
SCHEMBL14127680 0.80 DGAT1 (0.61) DGAT1KCNH2
SCHEMBL14127751 0.80 DGAT1 (0.61) DGAT1KCNH2
SCHEMBL19134107 0.80 FFAR4 (0.61) FFAR4FFAR1
SCHEMBL2559241 0.77 CYP2D6 (0.56) CYP3A4CYP2C9KCNH2
SCHEMBL20417178 0.76 LMNA (0.52) DGAT1KCNH2
SCHEMBL15073173 0.76 DGAT1 (0.57) FFAR4DGAT1CYP3A4CYP2C9KCNH2
SCHEMBL15058087 0.76 DGAT1 (0.67) FFAR4DGAT1CYP3A4CYP2C9KCNH2
SCHEMBL10146410 0.76 DGAT1 (0.76) FFAR4DGAT1CYP3A4CYP2C9KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012009217-A1 SPIROCYCLIC COMPOUNDS MERCK SHARP & DOHME CORP. (US) 2012-01-19 WO disclosed