SCHEMBL360849

SCHEMBL360849

Nc1cc(C(F)(F)F)ccc1NC(=O)c1cnc(Br)c(F)c1

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 5/20 0.49
HDAC1 Q13547 5/20 0.48
HDAC3 O15379 5/20 0.44
HDAC2 Q92769 4/20 0.44
CSF1R P07333 1/20 0.43
KIT P10721 1/20 0.43
NCOR2 Q9Y618 2/20 0.42
HDAC6 Q9UBN7 2/20 0.42
HSD17B10 Q99714 1/20 0.41
LIPE Q05469 1/20 0.41
CYP1A2 P05177 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14967989 0.88 PTGS1 (0.51) PTGS1HDAC1HDAC3HDAC2CSF1R
SCHEMBL1233684 0.80 KCNQ3 (0.60) PTGS1HDAC1LIPECYP1A2CYP2C19
SCHEMBL14453684 0.78 PTGS1 (0.61) PTGS1HDAC1HDAC3HDAC2
SCHEMBL27040039 0.77 PTGS1 (0.64) PTGS1HDAC1HDAC2CYP1A2CYP2C19
SCHEMBL1236023 0.75 PTGS1 (0.51) PTGS1HDAC1HDAC3HDAC2NCOR2
SCHEMBL3758034 0.74 PTGS1 (0.58) PTGS1HDAC1HDAC3HDAC2NCOR2
SCHEMBL23992191 0.73 HDAC3 (0.52) PTGS1HDAC1HDAC3HDAC2NCOR2
SCHEMBL30416650 0.73 HDAC3 (0.63) PTGS1HDAC1HDAC3HDAC2HDAC6
SCHEMBL15550450 0.73 HDAC1 (0.72) PTGS1HDAC1HDAC3HDAC2NCOR2
SCHEMBL22288985 0.72 KDM4E (0.53) HDAC1HDAC3HDAC2HDAC6CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012009217-A1 SPIROCYCLIC COMPOUNDS MERCK SHARP & DOHME CORP. (US) 2012-01-19 WO disclosed