SCHEMBL361732

SCHEMBL361732

Cc1ccccc1C(C/C(=N\O)c1ccc(=O)[nH]c1C)c1ccc(C(=O)NC(CO)CO)cc1

nearest known ligand 0.43

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 5/20 0.43
CTSA P10619 6/20 0.35
HSD17B2 P37059 1/20 0.35
SLC6A9 P48067 1/20 0.34
PAK4 O96013 3/20 0.34
TYMS P04818 1/20 0.33
MMP2 P08253 2/20 0.32
MMP9 P14780 2/20 0.32
MMP12 P39900 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL371107 0.85 GPBAR1 (0.42) GPBAR1CTSAHSD17B2SLC6A9
SCHEMBL15949284 0.84 GPBAR1 (0.60) GPBAR1CTSAHSD17B2
SCHEMBL370207 0.83 GPBAR1 (0.42) GPBAR1SLC6A9
SCHEMBL369130 0.79 GPBAR1 (0.49) GPBAR1CTSASLC6A9
SCHEMBL1389778 0.79 GPBAR1 (0.49) GPBAR1CTSASLC6A9
SCHEMBL1389775 0.79 GPBAR1 (0.49) GPBAR1CTSASLC6A9
SCHEMBL369898 0.75 GPBAR1 (0.42) GPBAR1CTSASLC6A9MMP2MMP9
SCHEMBL361767 0.73 GPBAR1 (0.47) GPBAR1CTSASLC6A9
SCHEMBL362542 0.73 GPBAR1 (0.47) GPBAR1CTSASLC6A9
SCHEMBL15949003 0.72 GPBAR1 (0.48) GPBAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed