SCHEMBL371107

SCHEMBL371107

Cc1ccccc1C(C/C(=N\O)c1ccc(=O)[nH]c1C)c1ccc(C(=O)NC2(CO)CC2)cc1

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 5/20 0.42
HSD17B2 P37059 1/20 0.33
MAPK8 P45983 1/20 0.32
SMN1; SMN2 Q16637 2/20 0.31
TP53 P04637 1/20 0.31
CTSA P10619 4/20 0.31
SLC6A9 P48067 1/20 0.31
KDM4E B2RXH2 1/20 0.31
MAPT P10636 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
EPHX2 P34913 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL361732 0.85 GPBAR1 (0.43) GPBAR1HSD17B2CTSASLC6A9
SCHEMBL364644 0.82 GPBAR1 (0.45) GPBAR1MAPK8SMN1; SMN2TP53CTSA
SCHEMBL15949284 0.82 GPBAR1 (0.60) GPBAR1HSD17B2CTSA
SCHEMBL371108 0.81 GPBAR1 (0.46) GPBAR1MAPK8SMN1; SMN2TP53MAPT
SCHEMBL1390109 0.81 GPBAR1 (0.46) GPBAR1MAPK8SMN1; SMN2TP53MAPT
SCHEMBL1390107 0.81 GPBAR1 (0.46) GPBAR1MAPK8SMN1; SMN2TP53MAPT
SCHEMBL370207 0.81 GPBAR1 (0.42) GPBAR1SLC6A9EPHX2
SCHEMBL362661 0.75 BRD4 (0.38) GPBAR1MAPK8SMN1; SMN2TP53CTSA
SCHEMBL1390479 0.74 GPBAR1 (0.37) GPBAR1MAPK8SMN1; SMN2TP53CTSA
SCHEMBL15949003 0.70 GPBAR1 (0.48) GPBAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed