SCHEMBL361844

SCHEMBL361844

Cc1cc(/C(CC(c2ccc(-c3ccc(C(=O)O)c(F)c3)cc2)c2ccccc2Cl)=N/O)c[nH]c1=O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 4/20 0.44
AXL P30530 1/20 0.35
ADRB1 P08588 1/20 0.34
ADRB3 P13945 1/20 0.34
BRD4 O60885 1/20 0.34
RARB P10826 3/20 0.33
RARA P10276 2/20 0.33
RARG P13631 1/20 0.33
S1PR1 P21453 1/20 0.33
S1PR3 Q99500 1/20 0.33
FFAR1 O14842 1/20 0.33
CTSA P10619 2/20 0.32
PRKAB2 O43741 3/20 0.32
PRKAG1 P54619 3/20 0.32
PRKAA2 P54646 3/20 0.32
PRKAA1 Q13131 3/20 0.32
PRKAG3 Q9UGI9 3/20 0.32
PRKAG2 Q9UGJ0 3/20 0.32
PRKAB1 Q9Y478 3/20 0.32
F9 P00740 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL362317 0.93 GPBAR1 (0.52) GPBAR1AXLADRB1ADRB3BRD4
SCHEMBL364504 0.92 GPBAR1 (0.40) GPBAR1BRD4FFAR1CTSAF9
SCHEMBL363296 0.91 GPBAR1 (0.38) GPBAR1ADRB1ADRB3BRD4RARB
SCHEMBL362646 0.91 GPBAR1 (0.38) GPBAR1ADRB1ADRB3BRD4RARB
SCHEMBL363787 0.91 GPBAR1 (0.38) GPBAR1ADRB1ADRB3BRD4RARB
SCHEMBL362527 0.89 GPBAR1 (0.55) GPBAR1ADRB1ADRB3BRD4CTSA
SCHEMBL364367 0.89 GPBAR1 (0.39) GPBAR1AXLADRB1ADRB3BRD4
SCHEMBL364998 0.89 GPBAR1 (0.39) GPBAR1AXLADRB1ADRB3BRD4
SCHEMBL363089 0.89 GPBAR1 (0.39) GPBAR1AXLADRB1ADRB3BRD4
SCHEMBL363245 0.85 GPBAR1 (0.43) GPBAR1AXLBRD4RARBRARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP claimed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO claimed
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed