SCHEMBL363245

SCHEMBL363245

Cc1ccccc1C(C/C(=N\O)c1c[nH]c(=O)c(C)c1)c1ccc(-c2ccc(C(=O)O)c(F)c2)cc1F

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 4/20 0.43
S1PR1 P21453 1/20 0.34
S1PR3 Q99500 1/20 0.34
FFAR1 O14842 1/20 0.34
CTSA P10619 5/20 0.33
RARB P10826 3/20 0.33
RARA P10276 2/20 0.33
AXL P30530 1/20 0.33
RARG P13631 1/20 0.33
MGLL Q99685 2/20 0.33
BRD4 O60885 1/20 0.33
PTGER4 P35408 2/20 0.32
CYP3A4 P08684 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL362317 0.92 GPBAR1 (0.52) GPBAR1S1PR1S1PR3FFAR1CTSA
SCHEMBL361842 0.92 GPBAR1 (0.51) GPBAR1FFAR1CTSABRD4PTGER4
SCHEMBL363216 0.92 GPBAR1 (0.39) GPBAR1FFAR1CTSABRD4CYP3A4
SCHEMBL363831 0.91 GPBAR1 (0.42) GPBAR1CTSABRD4
SCHEMBL363688 0.91 GPBAR1 (0.38) GPBAR1CTSABRD4CYP3A4
SCHEMBL364998 0.85 GPBAR1 (0.39) GPBAR1S1PR1S1PR3FFAR1RARB
SCHEMBL361844 0.85 GPBAR1 (0.44) GPBAR1S1PR1S1PR3FFAR1CTSA
SCHEMBL364367 0.85 GPBAR1 (0.39) GPBAR1S1PR1S1PR3FFAR1RARB
SCHEMBL363089 0.85 GPBAR1 (0.39) GPBAR1S1PR1S1PR3FFAR1RARB
SCHEMBL1390112 0.82 GPBAR1 (0.44) GPBAR1S1PR1S1PR3FFAR1CTSA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP claimed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO claimed
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed