SCHEMBL3622963

SCHEMBL3622963

CCOc1nc(NC2CCC(NC(=O)O)CC2)c(F)cc1C(N)=O

nearest known ligand 0.62

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 2/20 0.62
ROCK1 Q13464 1/20 0.62
SYK P43405 5/20 0.45
MAPK8 P45983 10/20 0.38
MAPK9 P45984 5/20 0.38
CDK1 P06493 1/20 0.38
CDK4 P11802 1/20 0.38
CCND1 P24385 1/20 0.38
CDK2 P24941 1/20 0.38
ALDH1A1 P00352 1/20 0.37
CSNK2A1 P68400 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3622961 1.00 ROCK2 (0.62) ROCK2ROCK1SYKMAPK8MAPK9
SCHEMBL12408592 0.89 ROCK2 (0.78) ROCK2ROCK1SYKMAPK8MAPK9
Hydrochloric Acid SCHEMBL1938755 0.88 ROCK2 (0.76) ROCK2ROCK1SYKMAPK8MAPK9
Hydrochloric Acid SCHEMBL1938754 0.88 ROCK2 (0.76) ROCK2ROCK1SYKMAPK8MAPK9
SCHEMBL3627381 0.88 ROCK2 (0.79) ROCK2ROCK1SYKMAPK8MAPK9
SCHEMBL3627383 0.88 ROCK2 (0.79) ROCK2ROCK1SYKMAPK8MAPK9
SCHEMBL3628622 0.88 ROCK2 (0.57) ROCK2ROCK1SYKMAPK8ALDH1A1
SCHEMBL3628618 0.88 ROCK2 (0.57) ROCK2ROCK1SYKMAPK8ALDH1A1
SCHEMBL3629563 0.87 ROCK2 (0.46) ROCK2ROCK1SYKMAPK8MAPK9
SCHEMBL3630680 0.87 ROCK2 (0.46) ROCK2ROCK1SYKMAPK8MAPK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010032875-A2 HETEROCYCLIC CARBOXAMIDE COMPOUNDS ASTELLAS PHARMA INC. (JP) 2010-03-25 WO disclosed