SCHEMBL362313

SCHEMBL362313

C/C(=N/O)[C@](c1ccc(N2CCC(CO)CC2)cc1)(c1ccnc(C)c1)c1ccccc1C

nearest known ligand 0.33

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ITGB2 P05107 2/20 0.33
ICAM1 P05362 2/20 0.33
ITGAL P20701 2/20 0.33
BRD4 O60885 1/20 0.33
PDE10A Q9Y233 2/20 0.33
LDHA P00338 1/20 0.32
LRRK2 Q5S007 2/20 0.31
RORC P51449 1/20 0.31
ITGB3 P05106 2/20 0.31
ITGB1 P05556 2/20 0.31
ITGAV P06756 2/20 0.31
ITGA2B P08514 2/20 0.31
ITGA5 P08648 2/20 0.31
ITGB5 P18084 2/20 0.31
WEE1 P30291 1/20 0.31
RXRA P19793 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL364429 0.89 LDHA (0.36) ITGB2ICAM1ITGALBRD4PDE10A
SCHEMBL362833 0.86 PSEN1 (0.38) BRD4
SCHEMBL365064 0.86 PSEN1 (0.38) BRD4
SCHEMBL362885 0.82
SCHEMBL363704 0.79
SCHEMBL364180 0.79 GPBAR1 (0.35)
SCHEMBL364263 0.78 GPBAR1 (0.31)
SCHEMBL363805 0.78 GPBAR1 (0.31)
SCHEMBL362830 0.78 TLR9 (0.38)
SCHEMBL364539 0.77 POLB (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP claimed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO claimed
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed