SCHEMBL3623951

SCHEMBL3623951

CC1CC(c2cn(S(=O)(=O)c3ccc4c(c3)N(C)CCO4)c3cccnc23)=CCN1

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PKM P14618 2/20 0.41
NPC1 O15118 1/20 0.41
PKLR P30613 1/20 0.41
RAB9A P51151 1/20 0.41
HTR6 P50406 12/20 0.39
HTR1A P08908 3/20 0.39
DRD2 P14416 3/20 0.39
HTR2A P28223 3/20 0.39
HTR7 P34969 3/20 0.39
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
DRD3 P35462 1/20 0.36
PPARG P37231 1/20 0.34
PPARD Q03181 1/20 0.34
PPARA Q07869 1/20 0.34
KMT2A Q03164 1/20 0.33
KLKB1 P03952 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3340203 0.86 HTR6 (0.54) HTR6HTR1ADRD2HTR2AHTR7
SCHEMBL3337575 0.83 HTR6 (0.51) PKMNPC1PKLRRAB9AHTR6
SCHEMBL3625114 0.81 NR3C2 (0.44) PKMRAB9AHTR6HTR1ADRD2
SCHEMBL3334361 0.81 HTR6 (0.53) HTR6HTR1ADRD2HTR2AHTR7
SCHEMBL3624153 0.80 HTR6 (0.43) HTR6HTR1ADRD2HTR2AHTR7
SCHEMBL3621987 0.79 HTR6 (0.46) PKMNPC1PKLRRAB9AHTR6
SCHEMBL3621695 0.79 HTR6 (0.42) HTR6HTR1ADRD2HTR2AHTR7
SCHEMBL3621648 0.79 HTR6 (0.39) HTR6HTR1ADRD2HTR2AHTR7
SCHEMBL3335906 0.78 HTR6 (0.50) HTR6HTR1ADRD2HTR2AHTR7
SCHEMBL3624061 0.76 AKR1C3 (0.46) RAB9AHTR6HTR1ADRD2HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2184990-A2 3' SUBSTITUTED COMPOUNDS HAVING 5-HT6 RECEPTOR AFFINITY Memory Pharmaceuticals Corporation (US) 2010-05-19 EP disclosed
WO-2009023844-A2 3' SUBSTITUTED COMPOUNDS HAVING 5-HT6 RECEPTOR AFFINITY MEMORY PHARMACEUTICALS CORPORATION (US) 2009-02-19 WO disclosed