SCHEMBL362609

SCHEMBL362609

N#Cc1cnn2cnc3ccccc3c12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 1/20 0.41
CDK2 P24941 1/20 0.41
KDM4E B2RXH2 5/20 0.39
MAP2K1 Q02750 2/20 0.36
RAF1 P04049 1/20 0.36
ALDH1A1 P00352 4/20 0.36
HPGD P15428 3/20 0.35
CLK4 Q9HAZ1 1/20 0.35
BMPR1B O00238 1/20 0.35
BMPR1A P36894 1/20 0.35
ACVR1B P36896 1/20 0.35
ACVRL1 P37023 1/20 0.35
ACVR1 Q04771 1/20 0.35
BMP4 P12644 1/20 0.35
MEN1 O00255 1/20 0.34
TP53 P04637 1/20 0.34
MAPT P10636 1/20 0.34
ALOX15 P16050 1/20 0.34
TSHR P16473 1/20 0.34
CASP1 P29466 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL362985 0.76 KDM4E (0.49) KDM4EALDH1A1HPGDBMP4TP53
SCHEMBL9138422 0.76 NCF1 (0.43) KDM4EALDH1A1HPGDBMP4CASP1
SCHEMBL11316779 0.70 FGFR1 (0.46) KDM4EALDH1A1MEN1MAPTTSHR
SCHEMBL4817117 0.68 KDM4E (0.39) LRRK2KDM4EMAP2K1RAF1ALDH1A1
SCHEMBL11315509 0.67 KMT2A (0.49) KDM4EALDH1A1HPGDMEN1TP53
SCHEMBL15452583 0.66 MKNK1 (0.46) LRRK2KDM4EMAP2K1RAF1MEN1
SCHEMBL828123 0.65 NCF1 (0.50) LRRK2KDM4EMAP2K1RAF1ALDH1A1
SCHEMBL29619912 0.65 NCF1 (0.50) LRRK2KDM4EMAP2K1RAF1ALDH1A1
SCHEMBL1164857 0.65 LRRK2 (0.54) LRRK2KDM4EMAP2K1RAF1ALDH1A1
SCHEMBL1346465 0.65 LRRK2 (0.54) LRRK2KDM4EMAP2K1RAF1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012007006-A1 TRIAZOLO- AND PYRAZOLOQUINAZOLINE DERIVATIVES AS PDE10A ENZYME INHIBITOR H. LUNDBECK A/S (DK) 2012-01-19 WO disclosed