SCHEMBL362915

SCHEMBL362915

CC(C)(C)OC(=O)n1nccc1B(O)O

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
FAAH O00519 1/20 0.38
ELANE P08246 1/20 0.36
BCHE P06276 1/20 0.36
POLB P06746 1/20 0.35
GPR119 Q8TDV5 5/20 0.33
USP2 O75604 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
MAPK1 P28482 1/20 0.33
USP30 Q70CQ3 1/20 0.33
ABCB1 P08183 1/20 0.32
SCD5 Q86SK9 1/20 0.32
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL693588 0.78 FAAH (0.41) FAAHELANEBCHEPOLBGPR119
SCHEMBL22951279 0.77 FAAH (0.40) FAAHELANEBCHEPOLBGPR119
SCHEMBL22501848 0.77 ELANE (0.44) FAAHELANEBCHEPOLBGPR119
SCHEMBL1864917 0.77 FAAH (0.40) FAAHELANEBCHEPOLBGPR119
SCHEMBL22233152 0.75 FAAH (0.39) FAAHELANEBCHEPOLBGPR119
SCHEMBL28739878 0.75 ELANE (0.42) FAAHELANEBCHEPOLBGPR119
SCHEMBL16630273 0.74 GABRA1 (0.40) FAAHELANEBCHEPOLBGPR119
SCHEMBL30879097 0.74 FAAH (0.41) FAAHELANEBCHEPOLBGPR119
SCHEMBL359804 0.73 FAAH (0.37) FAAHELANEBCHEMAPK1MEN1
SCHEMBL692934 0.73 FAAH (0.40) FAAHELANEBCHEPOLBGPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 61 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117756833-A Synthesis method of 1- (tert-butoxycarbonyl) pyrazole-5-boric acid 大连双硼医药化工有限公司 2024-03-26 CN claimed
EP-4652154-A1 NOVEL ALPK1 INHIBITORS Pyrotech (Beijing) Biotechnology Co., Ltd. (CN) 2025-11-26 EP disclosed
US-20250188070-A1 ANTIPROLIFERATION COMPOUNDS AND USES THEREOF VERTEX PHARMACEUTICALS INCORPORATED 2025-06-12 US disclosed
CN-112236428-B Antiproliferative compounds and uses thereof 默克专利股份有限公司 2025-04-01 CN disclosed
US-12195453-B2 Antiproliferation compounds and uses thereof MERCK PATENT GMBH (DE) 2025-01-14 US disclosed
US-20240368169-A1 SUBSTITUTED TRICYCLIC COMPOUNDS AS PARP INHIBITORS AND USE THEREOF IMPACT THERAPEUTICS (SHANGHAI), INC. (CN) 2024-11-07 US disclosed
WO-2024153225-A1 NOVEL ALPK1 INHIBITORS PYROTECH (BEIJING) BIOTECHNOLOGY CO., LTD. (CN) 2024-07-25 WO disclosed
EP-4392425-A1 SUBSTITUTED TRICYCLIC COMPOUNDS AS PARP INHIBITORS AND USE THEREOF Impact Therapeutics (Shanghai), Inc. (CN) 2024-07-03 EP disclosed
EP-4043460-B1 ANTIPROLIFERATION COMPOUNDS AND USES THEREOF MERCK PATENT GMBH (DE) 2024-06-05 EP disclosed
CN-117980307-A Substituted tricyclic compounds as PARP inhibitors and application thereof 上海瑛派药业有限公司 2024-05-03 CN disclosed
US-20140113901-A1 IMIDAZOPYRIDAZINES AS AKT KINASE INHIBITORS BAYER INTELLECTUAL PROPERTY GMBH (DE) 2014-04-24 US disclosed
EP-2694510-A1 IMIDAZOPYRIDAZINES AS AKT KINASE INHIBITORS Bayer Intellectual Property GmbH (DE) 2014-02-12 EP disclosed
US-20130310405-A1 SUBSTITUTED PYRIMIDO[1,2-B]INDAZOLES AND THEIR USE AS MODULATORS OF THE PI3K/AKT PATHWAY BAYER INTELLECTUAL PROPERTY GMBH (DE) 2013-11-21 US disclosed
WO-2013154878-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF INFINITY PHARMACEUTICALS, INC. (US) 2013-10-17 WO disclosed
US-20130267521-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF INTELLIKINE LLC (US) 2013-10-10 US disclosed
US-20130190332-A1 Substituted Imidazo[1,2-a]pyrimidines and -pyridines BAYER INTELLECTUAL PROPERTY GMBH (DE) 2013-07-25 US disclosed
EP-2593451-A2 SUBSTITUTED IMIDAZO[1,2-A]PYRIMIDINES AND -PYRIDINES Bayer Intellectual Property GmbH (DE) 2013-05-22 EP disclosed
WO-2013048214-A2 NOVEL HETEROCYCLIC DERIVATIVES AND THEIR USES C&C RESEARCH LABORATORIES (KR) 2013-04-04 WO disclosed
WO-2012136776-A1 IMIDAZOPYRIDAZINES AS AKT KINASE INHIBITORS BAYER INTELLECTUAL PROPERTY GMBH (DE) 2012-10-11 WO disclosed
WO-2012007345-A2 SUBSTITUTED IMIDAZO[1,2-A]PYRIMIDINES AND -PYRIDINES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2012-01-19 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240368169-A1 SUBSTITUTED TRICYCLIC COMPOUNDS AS PARP INHIBITORS AND USE THEREOF PARP1, PARP2, PARP11 FAAH 2196/4885ELANE 1838/4885BCHE 4111/4885
US-12195453-B2 Antiproliferation compounds and uses thereof MKI67, MCL1, CCNI FAAH 4482/4885ELANE 1800/4885BCHE 4496/4885
US-20250188070-A1 ANTIPROLIFERATION COMPOUNDS AND USES THEREOF MKI67, MCL1, CCNI FAAH 4482/4885ELANE 1800/4885BCHE 4496/4885
US-20130190332-A1 Substituted Imidazo[1,2-a]pyrimidines and -pyridines PIK3CA, PIK3CD, PIK3CB FAAH 4585/4885ELANE 4365/4885BCHE 4516/4885
US-20130267521-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF PIK3CA, PIK3CD, PIK3CB FAAH 2876/4885ELANE 1219/4885BCHE 1766/4885
US-20140113901-A1 IMIDAZOPYRIDAZINES AS AKT KINASE INHIBITORS PI4KA, PI4KB, PIK3CD FAAH 4684/4885ELANE 4425/4885BCHE 3182/4885
US-20130310405-A1 SUBSTITUTED PYRIMIDO[1,2-B]INDAZOLES AND THEIR USE AS MODULATORS OF THE PI3K/AKT PATHWAY PIK3CA, PIK3CD, PIK3CB FAAH 4714/4885ELANE 4523/4885BCHE 4438/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.