SCHEMBL362984

SCHEMBL362984

CC1CCNC(=O)N1C

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6021850 0.82 ALOX5 (0.32)
SCHEMBL22035389 0.79
SCHEMBL3044 0.75
SCHEMBL13574954 0.75
SCHEMBL27332822 0.71 AR (0.31)
SCHEMBL25653277 0.71 PIK3CD (0.31)
SCHEMBL14334701 0.70 MEN1 (0.33)
SCHEMBL8277266 0.70 P2RX7 (0.34)
SCHEMBL1260122 0.68 PER2 (0.44)
Phosphonic Acid SCHEMBL11341452 0.67 P2RX7 (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 259 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20160276056-A1 DISPERSIONS FOR NANOPLATELETS OF GRAPHENE-LIKE MATERIALS AND METHODS FOR PREPARING AND USING SAME GRAPHENE 3D LAB INC. (US) 2016-09-22 US claimed
EP-3047283-A1 SOLUTION FOR DISSOCIATING VITAMIN D FROM VITAMIN D-BINDING PROTEIN, ASSOCIATED DETECTION METHOD AND USE Biomérieux (FR) 2016-07-27 EP claimed
US-20150133569-A1 CARBON NANOTUBE SUSPENSIONS AND METHODS OF MAKING THE SAME CHEIL INDUSTRIES, INC. (KR) 2015-05-14 US claimed
EP-2866919-A1 AQUEOUS ALKANOLAMINE SOLUTION AND PROCESS FOR THE REMOVAL OF H2S FROM GASEOUS MIXTURES Dow Global Technologies LLC (US) 2015-05-06 EP claimed
US-20150087858-A1 CARBON NANOTUBE SUSPENSIONS AND METHODS OF MAKING THE SAME CHEIL INDUSTRIES INC. (KR) 2015-03-26 US claimed
WO-2015040319-A1 SOLUTION FOR DISSOCIATING VITAMIN D FROM VITAMIN D-BINDING PROTEIN, ASSOCIATED DETECTION METHOD AND USE bioMérieux (FR) 2015-03-26 WO claimed
WO-2014210584-A1 DISPERSIONS FOR NANOPLATELETS OF GRAPHENE-LIKE MATERIALS GRAPHENE 3D LAB INC. (US) 2014-12-31 WO claimed
WO-2014004020-A1 AQUEOUS ALKANOLAMINE SOLUTION AND PROCESS FOR THE REMOVAL OF H2S FROM GASEOUS MIXTURES DOW GLOBAL TECHNOLOGIES LLC (US) 2014-01-03 WO claimed
US-8148353-B2 Polymorphs of fluticasone furoate and process for preparation thereof PLUS CHEMICALS SA (CH) 2012-04-03 US claimed
US-20100130458-A1 Polymorphs of fluticasone furoate and process for preparation thereof PLUS CHEMICALS SA (CH) 2010-05-27 US claimed
US-6301038-B1 IN BUILDINGS AND AUTOMOBILES UNIVERSITY COLLEGE DUBLIN (IE) 2001-10-09 US claimed
EP-0958526-A1 ELECTROCHROMIC SYSTEM UNIVERSITY COLLEGE DUBLIN (IE) 1999-11-24 EP claimed
EP-0886804-A2 ELECTROCHROMIC OR PHOTOELECTROCHROMIC DEVICE Ecole Polytechnique Féderale de Lausanne (EPFL) (CH) 1998-12-30 EP claimed
EP-0882062-A1 METHOD OF PREPARING 21-ALKYLATED PREGNA-1,4,16-TRIEN-3,20-DIONES ALCON LABORATORIES, INC. (US) 1998-12-09 EP claimed
WO-1998035267-A1 ELECTROCHROMIC SYSTEM UNIVERSITY COLLEGE DUBLIN (IE) 1998-08-13 WO claimed
WO-1998018813-A1 METHOD OF PREPARING 21-ALKYLATED PREGNA-1,4,16-TRIEN-3,20-DIONES ALCON LABORATORIES, INC. (US) 1998-05-07 WO claimed
WO-1997035227-A2 ELECTROCHROMIC OR PHOTOELECTROCHROMIC DEVICE ECOLE POLYTECHNIQUE FEDERALE DE LAUSANNE (CH) 1997-09-25 WO claimed
US-5523269-A USING A COAL DERIVED MATERIAL ENERKOM (PROPRIETARY) LIMITED (ZA) 1996-06-04 US claimed
US-5340511-A Providing solution of coal-derived material in a solvent, adding polyethylene oxide, spinning ENERKOM (PROPRIETARY LIMITED (ZA) 1994-08-23 US claimed
EP-0371563-A1 Preparation of halofluorobenzenes DOWELANCO (US) 1990-06-06 EP claimed