Desmethoxyyangonin

Desmethoxyyangonin

SCHEMBL3630674

COc1cc(/C=C/c2ccccc2)oc(=O)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 1.00
HPGD P15428 5/20 1.00
SMN1; SMN2 Q16637 4/20 1.00
TP53 P04637 3/20 1.00
CYP3A4 P08684 2/20 1.00
MAPT P10636 5/20 0.82
HSD17B10 Q99714 2/20 0.82
CASP1 P29466 1/20 0.82
CASP7 P55210 1/20 0.82
HIF1A Q16665 1/20 0.64
TRPA1 O75762 1/20 0.56
KDM4E B2RXH2 4/20 0.52
MEN1 O00255 1/20 0.51
USP2 O75604 1/20 0.51
KMT2A Q03164 1/20 0.51
TRPV1 Q8NER1 1/20 0.51
MAOA P21397 2/20 0.48
MAOB P27338 2/20 0.48
NPC1 O15118 2/20 0.48
RAB9A P51151 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Desmethoxyyangonin SCHEMBL236641 1.00 ALDH1A1 (1.00) ALDH1A1HPGDSMN1; SMN2TP53CYP3A4
Yangonin SCHEMBL1393965 0.90 ALDH1A1 (1.00) ALDH1A1HPGDSMN1; SMN2TP53CYP3A4
Yangonin SCHEMBL5584097 0.90 ALDH1A1 (1.00) ALDH1A1HPGDSMN1; SMN2TP53CYP3A4
SCHEMBL9016266 0.86 MAPT (0.80) ALDH1A1HPGDSMN1; SMN2TP53CYP3A4
SCHEMBL9016268 0.86 MAPT (0.80) ALDH1A1HPGDSMN1; SMN2TP53CYP3A4
SCHEMBL9016241 0.82 HIF1A (0.78) ALDH1A1HPGDSMN1; SMN2TP53CYP3A4
SCHEMBL29584432 0.82 HIF1A (0.78) ALDH1A1HPGDSMN1; SMN2TP53CYP3A4
SCHEMBL9016238 0.82 HIF1A (0.78) ALDH1A1HPGDSMN1; SMN2TP53CYP3A4
SCHEMBL19665470 0.81 HIF1A (0.80) ALDH1A1HPGDSMN1; SMN2TP53CYP3A4
SCHEMBL19665468 0.81 HIF1A (0.80) ALDH1A1HPGDSMN1; SMN2TP53CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 45 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112353791-B Slip-derived therapeutic compounds and methods of use thereof 夸利蒂赫布丘蒂克斯公司 2025-02-25 CN disclosed
US-20240374519-A1 COMPOSITIONS FOR SUPPLEMENTING PRODUCTS WITH THERAPEUTIC AGENTS AND METHODS OF USE THEREOF DISRUPTION LABS, INC. (US) 2024-11-14 US disclosed
CN-118290377-A Extraction method of kavalactones for cosmetics 西安绿天生物技术有限公司 2024-07-05 CN disclosed
EP-4319722-A1 COMPOSITIONS FOR SUPPLEMENTING PRODUCTS WITH THERAPEUTIC AGENTS AND METHODS OF USE THEREOF Disruption Labs Inc. (US) 2024-02-14 EP disclosed
WO-2023194953-A1 COMPOSITIONS FOR SUPPLEMENTING PRODUCTS WITH THERAPEUTIC AGENTS AND METHODS OF USE THEREOF DISRUPTION LABS, INC. (US) 2023-10-12 WO disclosed
WO-2023150361-A1 KAVA COMPOSITIONS AND METHODS OF MAKING SAME Botanic Tonics, LLC (US) 2023-08-10 WO disclosed
US-20230233466-A1 COMPOSITIONS FOR SUPPLEMENTING PRODUCTS WITH THERAPEUTIC AGENTS AND METHODS OF USE THEREOF CORENHANCED TECHNOLOGIES LLC 2023-07-27 US disclosed
CN-116322732-A Compositions for supplementing products with therapeutic agents and methods of use thereof 迪斯拉普申实验室公司 2023-06-23 CN disclosed
WO-2023067509-A1 COMPOSITIONS FOR SUPPLEMENTING KOMBUCHA PRODUCTS WITH THERAPEUTIC AGENTS AND METHODS OF MAKING AND USE THEREOF DISRUPTION LABS, INC. (US) 2023-04-27 WO disclosed
EP-4168900-A1 COMPOSITIONS FOR SUPPLEMENTING PRODUCTS WITH THERAPEUTIC AGENTS AND METHODS OF USE THEREOF Disruption Labs Inc. (US) 2023-04-26 EP disclosed
US-7199152-B2 TNF-α production inhibitor comprising kavalactone as an active ingredient MEIJI DAIRIES CORPORATION (JP) 2007-04-03 US disclosed
US-7199152-B2 TNF-α production inhibitor comprising kavalactone as an active ingredient MEIJI DAIRIES CORPORATION (JP) 2007-04-03 US disclosed
US-20050069596-A1 Compositions and methods comprising kava and anti-anxiety compounds HERBALSCIENCE NUTRACEUTICALS, INC. 2005-03-31 US disclosed
US-20050037025-A1 Methods and compositions comprising kava and mate' or theobromine HERBALSCIENCE NUTRACEUTICALS, INC. 2005-02-17 US disclosed
EP-1032572-B1 PYRANONES, METHOD FOR THE PRODUCTION AND USE THEREOF SCHWABE WILLMAR GMBH & CO (DE) 2002-12-11 EP disclosed
US-6288109-B1 Pyranones, method for the production and use thereof DR. WILLMAR SCHWABE GMBH & CO. (DE) 2001-09-11 US disclosed
EP-1032572-A2 PYRANONES, METHOD FOR THE PRODUCTION AND USE THEREOF Dr. Willmar Schwabe GmbH & Co. (DE) 2000-09-06 EP disclosed
WO-1999025716-A9 PYRANONES, METHOD FOR THE PRODUCTION AND USE THEREOF SCHWABE WILLMAR GMBH & CO (DE) 1999-09-02 WO disclosed
WO-1999025716-A2 PYRANONES, METHOD FOR THE PRODUCTION AND USE THEREOF DR. WILLMAR SCHWABE GMBH & CO. (DE) 1999-05-27 WO disclosed
US-5585386-A MIXTURES FOR APPLICATION TO SKIN OR SCALP L'OREAL (FR) 1996-12-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050037025-A1 Methods and compositions comprising kava and mate' or theobromine ACHE, TES, KMT5C ALDH1A1 4389/4885HPGD 1621/4885SMN1; SMN2 1494/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.