SCHEMBL363976

SCHEMBL363976

Cc1cc(F)ccc1C(C/C(=N\O)c1c[nH]c(=O)c(C)c1)c1ccc(-c2ccc(C(=O)NCC(=O)O)cc2)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 3/20 0.41
EPHX2 P34913 2/20 0.37
SLC6A9 P48067 4/20 0.35
BRD4 O60885 1/20 0.34
EGLN1 Q9GZT9 2/20 0.34
ALDH1A1 P00352 2/20 0.33
MEN1 O00255 1/20 0.33
LMNA P02545 1/20 0.33
MAPT P10636 1/20 0.33
MAPK1 P28482 1/20 0.33
KMT2A Q03164 1/20 0.33
MCL1 Q07820 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
GART P22102 1/20 0.33
KDM4E B2RXH2 2/20 0.33
SLC6A5 Q9Y345 2/20 0.33
GCG P01275 1/20 0.33
MMP1 P03956 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
VEGFA P15692 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL363619 0.93 GPBAR1 (0.39) GPBAR1EPHX2SLC6A9BRD4ALDH1A1
SCHEMBL363289 0.90 GPBAR1 (0.41) GPBAR1EPHX2SLC6A9BRD4EGLN1
SCHEMBL363235 0.89 GPBAR1 (0.51) GPBAR1EPHX2BRD4MEN1MAPK1
SCHEMBL362350 0.86 GPBAR1 (0.48) GPBAR1EPHX2SLC6A9BRD4MAPT
SCHEMBL363293 0.85 GPBAR1 (0.39) GPBAR1BRD4ALDH1A1MEN1LMNA
SCHEMBL362551 0.85 GPBAR1 (0.38) GPBAR1ALDH1A1MEN1LMNAMAPT
SCHEMBL1390253 0.84 GPBAR1 (0.41) GPBAR1SLC6A9BRD4EGLN1KMT2A
SCHEMBL1390250 0.84 GPBAR1 (0.41) GPBAR1SLC6A9BRD4EGLN1KMT2A
SCHEMBL362887 0.83 GPBAR1 (0.39) GPBAR1BRD4EGLN1ALDH1A1MEN1
SCHEMBL362281 0.83 GPBAR1 (0.48) GPBAR1EPHX2BRD4LMNAMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP claimed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO claimed
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed