SCHEMBL363288

SCHEMBL363288

Cc1cc(Cl)ccc1C(C/C(=N\O)c1c[nH]c(=O)c(C)c1)c1ccc(-c2ccc(S(N)(=O)=O)cc2)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 2/20 0.39
CHRNA7 P36544 4/20 0.33
CA1 P00915 9/20 0.33
CA2 P00918 9/20 0.33
CA9 Q16790 9/20 0.33
CA12 O43570 5/20 0.33
CA14 Q9ULX7 2/20 0.33
CA4 P22748 3/20 0.33
KDM4E B2RXH2 1/20 0.32
MEN1 O00255 1/20 0.32
ALDH1A1 P00352 1/20 0.32
CYP1A2 P05177 1/20 0.32
POLB P06746 1/20 0.32
GAA P10253 1/20 0.32
CYP2D6 P10635 1/20 0.32
MAPT P10636 1/20 0.32
THRB P10828 1/20 0.32
CYP2C9 P11712 1/20 0.32
PKM P14618 1/20 0.32
MAPK1 P28482 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL365294 0.97 GPBAR1 (0.35) GPBAR1CHRNA7CA1CA2CA9
SCHEMBL363176 0.90 GPBAR1 (0.39) GPBAR1CHRNA7CA1CA2CA9
SCHEMBL363016 0.90 GPBAR1 (0.39) GPBAR1CHRNA7CA1CA2CA9
SCHEMBL364467 0.90 GPBAR1 (0.39) GPBAR1CHRNA7CA1CA2CA9
SCHEMBL362955 0.89 MGAM (0.38) CHRNA7CA1CA2CA9CA12
SCHEMBL363178 0.88 GPBAR1 (0.51) GPBAR1MEN1CYP1A2POLBGAA
SCHEMBL362796 0.85 GPBAR1 (0.39) GPBAR1KDM4EGAAMAPTKMT2A
SCHEMBL365274 0.85 GPBAR1 (0.46) GPBAR1MEN1CYP1A2POLBGAA
SCHEMBL361734 0.83 GPBAR1 (0.34) GPBAR1KDM4EMEN1KMT2AEP300
SCHEMBL12505651 0.83 GPBAR1 (0.35) GPBAR1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed