Phenylbutazone

Phenylbutazone

SCHEMBL3632

CCCCC1C(=O)N(c2ccccc2)N(c2ccccc2)C1=O

nearest known ligand 0.82

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

PTGS1PTGS2

The experimentally established mechanism targets of Phenylbutazone. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 known ✓ P23219 2/20 0.82
RAB9A P51151 3/20 0.82
ALDH1A1 P00352 2/20 0.82
CYP3A4 P08684 2/20 0.82
LMNA P02545 2/20 0.82
CYP1A2 P05177 2/20 0.82
CYP2C9 P11712 2/20 0.82
CYP2C19 P33261 2/20 0.82
MAPK1 P28482 1/20 0.82
TP53 P04637 1/20 0.82
MAPT P10636 1/20 0.82
HPGD P15428 1/20 0.82
NAPRT Q6XQN6 1/20 0.82
ABCB11 O95342 1/20 0.53
GRM2 Q14416 5/20 0.48
KDM4E B2RXH2 1/20 0.46
PKM P14618 1/20 0.46
SMN1; SMN2 Q16637 2/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Phenylbutazone SCHEMBL8005041 1.00 RAB9A (0.82) RAB9AALDH1A1CYP3A4LMNAPTGS1
Phenylbutazone SCHEMBL2122724 0.98 RAB9A (0.80) RAB9AALDH1A1CYP3A4LMNAPTGS1
Phenylbutazone SCHEMBL21694456 0.98 RAB9A (0.80) RAB9AALDH1A1CYP3A4LMNAPTGS1
Phenylbutazone SCHEMBL2874252 0.98 RAB9A (0.80) RAB9AALDH1A1CYP3A4LMNAPTGS1
Phenylbutazone SCHEMBL7715162 0.98 RAB9A (0.80) RAB9AALDH1A1CYP3A4LMNAPTGS1
Phenylbutazone SCHEMBL10913190 0.98 RAB9A (0.80) RAB9AALDH1A1CYP3A4LMNAPTGS1
SCHEMBL29489697 0.93 ALDH1A1 (0.73) RAB9AALDH1A1CYP3A4LMNAPTGS1
Phenylbutazone SCHEMBL11269971 0.92 ALDH1A1 (0.72) RAB9AALDH1A1CYP3A4LMNAPTGS1
Oxyphenbutazone Anhydrous SCHEMBL25857 0.91 LMNA (1.00) RAB9AALDH1A1CYP3A4LMNAPTGS1
Oxyphenbutazone Anhydrous SCHEMBL25856 0.91 LMNA (1.00) RAB9AALDH1A1CYP3A4LMNAPTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 62836 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4747263-A1 LIPID NANOPARTICLES AND USES THEREOF University of Connecticut (US) 2026-05-27 EP claimed
CN-121856715-B Method for judging ground fault of power distribution network and centralized protection measurement and control device 珠海菲森电力科技有限公司 2026-05-22 CN claimed
US-20260139030-A1 CHIMERIC PROTEINS FOR TREATING CUTANEOUS INFLAMMATION SHATTUCK LABS INC (US) 2026-05-21 US claimed
EP-4744679-A1 USE OF POLYLACTIC ACID AND COPOLYMER THEREOF IN PREPARATION OF DRUGS FOR PROMOTING TENDON/LIGAMENT GROWTH Changchun Sinobiomaterials Co., Ltd. (CN) 2026-05-20 EP claimed
CN-121580084-B Concrete pouring process monitoring method and system based on multi-source data 中国建筑第八工程局有限公司 2026-05-19 CN claimed
CN-116449143-B Relay protection device action time evaluation method and system based on machine learning algorithm 中国电力科学研究院有限公司 2026-05-19 CN claimed
CN-119864772-B Single-phase earth fault control method and system 国网浙江省电力有限公司瑞安市供电公司 2026-05-15 CN claimed
US-20260132404-A1 MODIFIED OLIGONUCLEOTIDES AND DOUBLE-STRANDED RNAS ALNYLAM PHARMACEUTICALS, INC. (US) 2026-05-14 US claimed
US-20260130928-A1 COMBINATION OF AKR1C3 ACTIVATED ANTICANCER PRODRUG COMPOUND AND ANALGESIC DRUG FOR TREATING CANCER PATIENTS ACCOMPANIED BY PAIN ASCENTAWITS PHARMACEUTICALS LTD (CN) 2026-05-14 US claimed
CN-122026283-A Longitudinal impedance differential protection method 华中科技大学 2026-05-12 CN claimed
WO-1980000661-A1 PHARMACEUTICAL PREPARATIONS CROFT J (NZ) 1980-04-17 WO claimed
EP-0010061-A1 Pharmaceutical preparations containing a mollusc extract Mc Farlane, Stuart John (NZ) 1980-04-16 EP claimed
US-4198402-A TO REDUCE ULCER-LESION FORMATION RICHTER GEDEON VEGYESZETI GYAR RT. (HU) 1980-04-15 US claimed
US-4175119-A Composition and method to prevent accidental and intentional overdosage with psychoactive drugs PORTER GARRY L 1979-11-20 US claimed
US-4169147-A Novel transient pro-drug forms of phenylbutazone and oxyphenbutazone in compositions and methods of use INTERX RESEARCH CORPORATION (US) 1979-09-25 US claimed
US-4168308-A Composition for enhancing the administration of pharmacologically active agents APOTEKSVARUCENTRALEN VITRUM AB (SE) 1979-09-18 US claimed
US-4151292-A ANTIINFLAMMATORY SIDE EFFECT INHIBITION USING CHROMENE DERIVATIVES, GASTROINTESTINAL DISORDERS FISONS LIMITED (GB) 1979-04-24 US claimed
US-4016268-A CO-ADMINISTERING A BISMUTH SUBSALICYLATE AND AN ANTIINFLAMMATORY AGENT MORTON-NORWICH PRODUCTS, INC. (US) 1977-04-05 US claimed
US-4004002-A PREVENT GASTRIC IRRITATION A. H. ROBINS COMPANY, INCORPORATED (US) 1977-01-18 US claimed
US-3993767-A ANTIINFLAMMATORY AGENTS A. H. ROBINS COMPANY, INCORPORATED (US) 1976-11-23 US claimed