SCHEMBL363831

SCHEMBL363831

Cc1ccccc1C(C/C(=N\O)c1c[nH]c(=O)c(C)c1)c1ccc(-c2ccccc2C(=O)O)cc1F

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 3/20 0.42
CTSA P10619 8/20 0.35
DHODH Q02127 1/20 0.34
LTB4R2 Q9NPC1 1/20 0.34
PPARG P37231 3/20 0.34
NR1I2 O75469 1/20 0.33
CYP2C9 P11712 1/20 0.33
IDO1 P14902 1/20 0.33
MCL1 Q07820 1/20 0.33
BRS3 P32247 1/20 0.32
BRD4 O60885 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL363245 0.91 GPBAR1 (0.43) GPBAR1CTSABRD4
SCHEMBL361842 0.89 GPBAR1 (0.51) GPBAR1CTSABRD4
SCHEMBL363216 0.85 GPBAR1 (0.39) GPBAR1CTSABRD4
SCHEMBL363688 0.84 GPBAR1 (0.38) GPBAR1CTSABRD4
SCHEMBL362317 0.84 GPBAR1 (0.52) GPBAR1CTSADHODHBRD4
SCHEMBL1390089 0.83 GPBAR1 (0.43) GPBAR1CTSALTB4R2PPARGNR1I2
SCHEMBL1390087 0.83 GPBAR1 (0.43) GPBAR1CTSALTB4R2PPARGNR1I2
SCHEMBL15949190 0.82 GPBAR1 (0.39) GPBAR1CTSADHODHLTB4R2PPARG
SCHEMBL362892 0.80 GPBAR1 (0.39) GPBAR1CTSAMCL1
SCHEMBL363623 0.80 GPBAR1 (0.39) GPBAR1PPARGCYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP claimed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO claimed
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed