SCHEMBL364313

SCHEMBL364313

Cc1cc(/C(CC(c2ccc(-c3ccc(CC#N)cc3)cc2)c2ccc(Cl)cc2F)=N/O)c[nH]c1=O

nearest known ligand 0.36

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
S1PR3 Q99500 3/20 0.36
S1PR1 P21453 1/20 0.36
GPBAR1 Q8TDU6 3/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL362367 0.89 GPBAR1 (0.38) S1PR3S1PR1GPBAR1
SCHEMBL364696 0.89 GPBAR1 (0.38) S1PR3S1PR1GPBAR1
SCHEMBL363327 0.89 GPBAR1 (0.38) S1PR3S1PR1GPBAR1
SCHEMBL361680 0.88 GPBAR1 (0.47) S1PR3S1PR1GPBAR1
SCHEMBL364367 0.86 GPBAR1 (0.39) S1PR3S1PR1GPBAR1
SCHEMBL363089 0.86 GPBAR1 (0.39) S1PR3S1PR1GPBAR1
SCHEMBL364998 0.86 GPBAR1 (0.39) S1PR3S1PR1GPBAR1
SCHEMBL363248 0.83 GPBAR1 (0.41) S1PR3S1PR1GPBAR1
SCHEMBL363638 0.83 GPBAR1 (0.41) S1PR3S1PR1GPBAR1
SCHEMBL363277 0.83 GPBAR1 (0.41) S1PR3S1PR1GPBAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP claimed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO claimed
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed