SCHEMBL3633273

SCHEMBL3633273

COc1cc(N)ccc1-c1ncc[nH]1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMPD3 Q9NY59 1/20 0.50
P2RX3 P56373 1/20 0.47
P2RX2 Q9UBL9 1/20 0.47
IMPDH2 P12268 1/20 0.47
IMPDH1 P20839 1/20 0.47
CDK4 P11802 1/20 0.44
CCNA2 P20248 1/20 0.44
CCND1 P24385 1/20 0.44
CDK2 P24941 1/20 0.44
CCND3 P30281 1/20 0.44
GAA P10253 2/20 0.42
MAPT P10636 2/20 0.42
KDM4E B2RXH2 2/20 0.42
TSHR P16473 1/20 0.42
MAPK1 P28482 1/20 0.42
HTT P42858 1/20 0.42
MC4R P32245 2/20 0.41
MAP3K11 Q16584 1/20 0.40
PDE7A Q13946 4/20 0.39
ALDH1A1 P00352 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6003238 0.82 PDE2A (0.55) SMPD3CDK4CCNA2CCND1CDK2
SCHEMBL15651168 0.78 NISCH (0.46) SMPD3GAAMAPTKDM4EALDH1A1
SCHEMBL3403152 0.78 ADRA1A (0.54) SMPD3GAAMC4RALDH1A1TUBB4A
SCHEMBL29360270 0.78 ADRA1A (0.54) SMPD3GAAMC4RALDH1A1TUBB4A
SCHEMBL5248703 0.78 CSNK1A1 (0.44) SMPD3GAAMAPTKDM4EALDH1A1
SCHEMBL3642126 0.77 SMPD3 (0.47) SMPD3P2RX3P2RX2CDK4CCNA2
SCHEMBL347390 0.76 MAPT (0.59) IMPDH2IMPDH1GAAMAPTKDM4E
SCHEMBL30839714 0.76 MAPT (0.59) IMPDH2IMPDH1GAAMAPTKDM4E
SCHEMBL32667989 0.76 CSNK1A1 (0.42) SMPD3GAAMAPTKDM4ETSHR
SCHEMBL8539151 0.76 CSNK1A1 (0.46) SMPD3GAAMAPTKDM4ETSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2155740-A1 HETARYLANILINES AS MODULATORS FOR AMYLOID BETA F. Hoffmann-Roche AG (CH) 2010-02-24 EP disclosed
WO-2008138753-A1 HETARYLANILINES AS MODULATORS FOR AMYLOID BETA F. HOFFMANN-LA ROCHE AG (CH) 2008-11-20 WO disclosed