SCHEMBL3633987

SCHEMBL3633987

Cc1cc2cc(Br)cc(C=O)c2[nH]1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 5/20 0.40
GRIA1 P42261 1/20 0.34
GRIA2 P42262 1/20 0.34
GRIA3 P42263 1/20 0.34
GRIA4 P48058 1/20 0.34
PIM3 Q86V86 2/20 0.33
ALDH1A1 P00352 2/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2C19 P33261 1/20 0.32
PIM1 P11309 1/20 0.32
HPGD P15428 2/20 0.32
CYP2A6 P11509 1/20 0.32
LMNA P02545 1/20 0.32
PRKDC P78527 1/20 0.32
KDM4E B2RXH2 3/20 0.31
GAA P10253 2/20 0.31
MAPT P10636 1/20 0.31
HTT P42858 2/20 0.30
SMN1; SMN2 Q16637 2/20 0.30
TDP1 Q9NUW8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12037745 0.74 KDM4E (0.42) ERN1GRIA1GRIA2GRIA3GRIA4
SCHEMBL28796378 0.73 CYP2A6 (0.37) HPGDCYP2A6LMNA
SCHEMBL29267034 0.73 IDO1 (0.36) PIM1HPGDLMNA
SCHEMBL30993119 0.70 CYP2A6 (0.41) ERN1PIM3PIM1CYP2A6
SCHEMBL28796435 0.70 ERN1 (0.41) ERN1ALDH1A1CYP1A2MAPTHTT
SCHEMBL31698302 0.69 NOS1 (0.42) ERN1ALDH1A1CYP1A2CYP2C19HPGD
SCHEMBL3636860 0.69 CYP19A1 (0.38) GRIA1GRIA2GRIA3GRIA4KDM4E
SCHEMBL28356912 0.68 PIM3 (0.41) ERN1GRIA1GRIA2GRIA3GRIA4
SCHEMBL29635192 0.66 NPY5R (0.43) ALDH1A1PIM1GAAMAPTHTT
SCHEMBL28796377 0.66 NPY5R (0.43) ALDH1A1PIM1GAAMAPTHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2152674-A1 BENZIMIDAZOLONE CHYMASE INHIBITORS Boehringer Ingelheim International GmbH (DE) 2010-02-17 EP disclosed
WO-2008147697-A1 BENZIMIDAZOLONE CHYMASE INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-12-04 WO disclosed