SCHEMBL28796378

SCHEMBL28796378

Cc1cc2cc(Br)cc(N)c2[nH]1

nearest known ligand 0.37

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.37
KEAP1 Q14145 1/20 0.37
MAP4K1 Q92918 1/20 0.32
IDO1 P14902 1/20 0.32
TDO2 P48775 1/20 0.32
CYP3A4 P08684 1/20 0.30
TSHR P16473 1/20 0.30
MAPK1 P28482 1/20 0.30
LMNA P02545 1/20 0.30
HPGD P15428 1/20 0.30
PARP1 P09874 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29267034 0.76 IDO1 (0.36) IDO1LMNAHPGD
SCHEMBL31078313 0.76 HRH4 (0.46) CYP2A6KEAP1MAP4K1CYP3A4TSHR
SCHEMBL3633987 0.73 ERN1 (0.40) CYP2A6LMNAHPGD
SCHEMBL3636860 0.72 CYP19A1 (0.38)
SCHEMBL25686336 0.72 ALDH1A1 (0.30)
SCHEMBL28359192 0.71 PDE4A (0.39) CYP2A6KEAP1LMNAHPGD
SCHEMBL6194760 0.69 PARP1 (0.46) CYP2A6KEAP1CYP3A4TSHRLMNA
SCHEMBL28796435 0.69 ERN1 (0.41)
SCHEMBL29635192 0.68 NPY5R (0.43)
SCHEMBL28796377 0.68 NPY5R (0.43)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113248472-B Anti-osteoporosis compound and derivative thereof, pharmaceutical composition, preparation method and application 中国药科大学 2022-06-28 CN disclosed
CN-113248472-A Anti-osteoporosis compound and derivative thereof, pharmaceutical composition, preparation method and application 中国药科大学 2021-08-13 CN disclosed