SCHEMBL3634306

SCHEMBL3634306

COc1ccc(Cn2nc(C(F)(F)F)cc2[C](C)c2cc(C(F)(F)F)n[nH]2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
ALDH1A1 P00352 2/20 0.38
F10 P00742 1/20 0.38
FABP4 P15090 2/20 0.38
GAA P10253 1/20 0.38
RECQL P46063 1/20 0.38
PTGS1 P23219 3/20 0.37
PTGS2 P35354 3/20 0.37
GRIN1 Q05586 1/20 0.37
GRIN2B Q13224 1/20 0.37
MAPT P10636 2/20 0.37
NPSR1 Q6W5P4 2/20 0.37
MAPK1 P28482 1/20 0.37
AKR1C3 P42330 1/20 0.37
TP53 P04637 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
TSHR P16473 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2688186 0.78 GRN (0.57) ALDH1A1F10GAARECQLMAPT
SCHEMBL14549306 0.78 ALDH1A1 (0.63) ALDH1A1F10GAARECQLMAPT
SCHEMBL4070158 0.78 ALDH1A1 (0.47) ALDH1A1F10GAARECQLMAPT
SCHEMBL3634308 0.75 FABP4 (0.39) KDM4ESMN1; SMN2FABP4PTGS1PTGS2
SCHEMBL1197409 0.74 KDM4E (0.52) KDM4ESMN1; SMN2ALDH1A1GAAPTGS1
SCHEMBL1197408 0.74 PTGS2 (0.50) FABP4PTGS1PTGS2GRIN1GRIN2B
Pivalate SCHEMBL27592717 0.73 MAPT (0.47) ALDH1A1F10GAARECQLMAPT
SCHEMBL287956 0.71 PTGS2 (0.44) FABP4PTGS1PTGS2GRIN1GRIN2B
SCHEMBL27977409 0.71 PTGS2 (0.44) SMN1; SMN2FABP4PTGS1PTGS2GRIN1
SCHEMBL2686357 0.68 AKR1C3 (0.42) KDM4ESMN1; SMN2ALDH1A1MAPTAKR1C3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2152664-A1 DIPEPTIDE ANALOGS AS COAGULATION FACTOR INHIBITORS Brystol-Myers Squibb Company (US) 2010-02-17 EP disclosed
WO-2008157162-A1 DIPEPTIDE ANALOGS AS COAGULATION FACTOR INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2008-12-24 WO disclosed