SCHEMBL3634758

SCHEMBL3634758

CCOC(=O)n1c(C(=O)O)cc2cc(OCCSC)ccc21

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SRD5A2 P31213 1/20 0.44
KDM4E B2RXH2 2/20 0.41
ALDH1A1 P00352 1/20 0.41
HPGD P15428 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
HSD17B10 Q99714 1/20 0.41
MAOA P21397 1/20 0.40
PLA2G4A P47712 6/20 0.39
KMT2A Q03164 2/20 0.39
MEN1 O00255 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
GFER P55789 1/20 0.39
MCL1 Q07820 1/20 0.39
LTB4R Q15722 1/20 0.38
LTB4R2 Q9NPC1 1/20 0.38
AR P10275 1/20 0.37
ADRB3 P13945 1/20 0.37
MAPT P10636 2/20 0.36
LMNA P02545 1/20 0.36
CCR2 P41597 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13560511 0.88 SRD5A2 (0.40) SRD5A2KDM4EALDH1A1HPGDSMN1; SMN2
SCHEMBL3634756 0.85 MAOA (0.45) SRD5A2KDM4EALDH1A1HPGDSMN1; SMN2
SCHEMBL3027681 0.83 NR1H2 (0.42) SRD5A2KDM4EHPGDSMN1; SMN2HSD17B10
SCHEMBL13560478 0.83 SRD5A2 (0.40) SRD5A2KDM4EALDH1A1HPGDSMN1; SMN2
SCHEMBL3639124 0.81 SRD5A2 (0.69) SRD5A2KDM4EALDH1A1HPGDHSD17B10
SCHEMBL13560509 0.80 MAOA (0.35) SRD5A2KDM4EMAOAKMT2AMEN1
SCHEMBL3023791 0.78 MAOA (0.43) HPGDMAOAKMT2AMEN1TDP1
SCHEMBL3637426 0.76 ABCB11 (0.45) SRD5A2KDM4EALDH1A1HPGDSMN1; SMN2
SCHEMBL3675353 0.76 KDM4E (0.42) SRD5A2KDM4EALDH1A1HPGDSMN1; SMN2
SCHEMBL13560475 0.75 MAOA (0.37) SRD5A2MAOAMCL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2166856-A1 CHEMICAL COMPOUNDS GlaxoSmithKline LLC (US) 2010-03-31 EP disclosed
WO-2008154271-A1 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2008-12-18 WO disclosed