SCHEMBL3675353

SCHEMBL3675353

CCOC(=O)n1c(C(=O)O)cc2cc(OS(=O)(=O)C(F)(F)F)ccc21

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.42
ALDH1A1 P00352 2/20 0.42
HPGD P15428 2/20 0.42
HSD17B10 Q99714 2/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
GFER P55789 1/20 0.40
SRD5A2 P31213 1/20 0.40
HSD11B1 P28845 1/20 0.38
CCR2 P41597 2/20 0.36
NR1H2 P55055 1/20 0.36
DRD2 P14416 1/20 0.36
HTR1D P28221 1/20 0.36
DRD3 P35462 1/20 0.36
PLA2G4A P47712 2/20 0.36
NTRK1 P04629 1/20 0.36
ADORA1 P30542 1/20 0.36
ABCB11 O95342 1/20 0.35
LGALS8 O00214 1/20 0.35
LGALS3 P17931 1/20 0.35
MEN1 O00255 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3675346 0.85 NOD2 (0.43) KDM4EALDH1A1HPGDHSD17B10SMN1; SMN2
SCHEMBL2813774 0.85 NOD2 (0.40) ALDH1A1HPGDHSD11B1NR1H2ADORA1
SCHEMBL3637426 0.77 ABCB11 (0.45) KDM4EALDH1A1HPGDHSD17B10SMN1; SMN2
SCHEMBL3639124 0.77 SRD5A2 (0.69) KDM4EALDH1A1HPGDHSD17B10SRD5A2
SCHEMBL3634758 0.76 SRD5A2 (0.44) KDM4EALDH1A1HPGDHSD17B10SMN1; SMN2
SCHEMBL1460272 0.76 ALDH1A1 (0.35) ALDH1A1HPGDHSD17B10SMN1; SMN2HSD11B1
SCHEMBL11890112 0.74 NR1H2 (0.43) ALDH1A1SMN1; SMN2NR1H2NTRK1MEN1
SCHEMBL5865527 0.73 STS (0.52) KDM4EALDH1A1HPGDHSD17B10SMN1; SMN2
SCHEMBL10173126 0.73 MAPT (0.41) ALDH1A1HPGDSMN1; SMN2MEN1KMT2A
SCHEMBL3639293 0.72 MMP13 (0.47) KDM4EALDH1A1HSD17B10SMN1; SMN2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2170072-A1 FARNESOID X RECEPTOR AGONISTS GlaxoSmithKline LLC (US) 2010-04-07 EP disclosed
WO-2008157270-A1 FARNESOID X RECEPTOR AGONISTS SMITHKLINE BEECHAM CORPORATION (US) 2008-12-24 WO disclosed