SCHEMBL3635401

SCHEMBL3635401

Cc1ccc(C(C(=O)O)N2CCN(C)CC2)c(C)n1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MC4R P32245 2/20 0.37
SLC1A2 P43004 1/20 0.36
HTR3E A5X5Y0 1/20 0.36
HTR3B O95264 1/20 0.36
HTR3A P46098 1/20 0.36
HTR3D Q70Z44 1/20 0.36
HTR3C Q8WXA8 1/20 0.36
LMNA P02545 1/20 0.36
CHRM2 P08172 1/20 0.35
CHRM4 P08173 1/20 0.35
CHRM5 P08912 1/20 0.35
ADRA2A P08913 1/20 0.35
ADORA3 P0DMS8 1/20 0.35
CYP2D6 P10635 1/20 0.35
CHRM1 P11229 1/20 0.35
CHRM3 P20309 1/20 0.35
DRD1 P21728 1/20 0.35
ADRA1D P25100 1/20 0.35
HTR2A P28223 1/20 0.35
HTR2C P28335 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13044650 0.84 MC4R (0.42) MC4ROPRM1KCNH2GAAOXTR
SCHEMBL3635298 0.79 SLC1A2 (0.42) SLC1A2
SCHEMBL3633189 0.77 HTR3E (0.45) MC4RSLC1A2HTR3EHTR3BHTR3A
SCHEMBL13984355 0.75 MC4R (0.49) MC4RSLC1A2LMNACHRM2CHRM4
SCHEMBL3638763 0.74 SLC1A2 (0.46) MC4RSLC1A2LMNACHRM2CHRM4
SCHEMBL13044372 0.74 GHSR (0.55) MC4RLMNACHRM2CHRM4CHRM5
Hydrochloric Acid SCHEMBL3639303 0.74 MC4R (0.48) MC4RLMNACHRM2CHRM4CHRM5
SCHEMBL3730182 0.73 GHSR (0.43) MC4RLMNAOXTRKDM4EGHSR
SCHEMBL3750634 0.73 GHSR (0.69) LMNAKDM4EALDH1A1GHSRMEN1
Hydrochloric Acid SCHEMBL3636742 0.72 GHSR (0.54) MC4RLMNACHRM2CHRM4CHRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2167466-A1 N-PHENYL HYDRAZIDES AS MODULATORS OF THE GHRELIN RECEPTOR Glaxo Group Limited (GB) 2010-03-31 EP disclosed
WO-2008148853-A1 N-PHENYL HYDRAZIDES AS MODULATORS OF THE GHRELIN RECEPTOR GLAXO GROUP LIMITED (GB) 2008-12-11 WO disclosed