SCHEMBL3635830

SCHEMBL3635830

CCNC(=O)N(C)C1CCN(c2ccc(C(N)=O)cc2)CC1

nearest known ligand 0.48

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 1/20 0.48
CHRNA10 Q9GZZ6 1/20 0.48
CHRNA9 Q9UGM1 1/20 0.48
NPY5R Q15761 12/20 0.45
GPR119 Q8TDV5 1/20 0.45
MCHR1 Q99705 2/20 0.43
USP2 O75604 1/20 0.41
SYK P43405 1/20 0.41
HRH3 Q9Y5N1 1/20 0.40
CHRM4 P08173 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3635452 0.91 CHRNA10 (0.46) CHRNA7CHRNA10CHRNA9NPY5RGPR119
SCHEMBL3636419 0.88 NPY5R (0.49) NPY5R
SCHEMBL3812349 0.78 NPY5R (0.47) CHRNA10CHRNA9NPY5RCHRM4
SCHEMBL2636306 0.75 MCHR1 (0.58) CHRNA7CHRNA10CHRNA9GPR119MCHR1
SCHEMBL4287740 0.75 MCHR1 (0.58) CHRNA7CHRNA10CHRNA9GPR119MCHR1
SCHEMBL2636123 0.74 MCHR1 (0.61) CHRNA7CHRNA10CHRNA9GPR119MCHR1
SCHEMBL16130769 0.72 USP2 (0.73) CHRNA7CHRNA10CHRNA9GPR119USP2
SCHEMBL3631885 0.72 GPR119 (0.53) CHRNA7CHRNA10CHRNA9GPR119MCHR1
SCHEMBL970988 0.72 ATM (0.39) NPY5R
SCHEMBL19658498 0.71 NPY5R (0.50) NPY5RGPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2155687-A1 DIACYLGLYCEROL ACYLTRANSFERASE INHIBITORS Via Pharmaceuticals, Inc. (US) 2010-02-24 EP disclosed
US-20090170864-A1 Diacylglycerol Acyltransferase Inhibitors MADRIGAL PHARMACEUTICALS, INC. 2009-07-02 US disclosed
US-20090105273-A1 Diacylglycerol Acyltransferase Inhibitors MADRIGAL PHARMACEUTICALS, INC. 2009-04-23 US disclosed
US-20090099201-A1 Diacylglycerol Acyltransferase Inhibitors VIA PHARMACEUTICALS, INC. 2009-04-16 US disclosed
US-20090093497-A1 Diacylglycerol Acyltransferase Inhibitors MADRIGAL PHARMACEUTICALS, INC. 2009-04-09 US disclosed
WO-2008141976-A1 DIACYLGLYCEROL ACYLTRANSFERASE INHIBITORS VIA PHARMACEUTICALS, INC. (US) 2008-11-27 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090093497-A1 Diacylglycerol Acyltransferase Inhibitors DGAT2, DGAT1, LCAT CHRNA7 4349/4885CHRNA10 4368/4885CHRNA9 4295/4885
US-20090170864-A1 Diacylglycerol Acyltransferase Inhibitors DGAT2, DGAT1, LCAT CHRNA7 4349/4885CHRNA10 4368/4885CHRNA9 4295/4885
US-20090099201-A1 Diacylglycerol Acyltransferase Inhibitors DGAT2, DGAT1, LCAT CHRNA7 4349/4885CHRNA10 4368/4885CHRNA9 4295/4885
US-20090105273-A1 Diacylglycerol Acyltransferase Inhibitors DGAT2, DGAT1, LCAT CHRNA7 4349/4885CHRNA10 4368/4885CHRNA9 4295/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.