SCHEMBL363585

SCHEMBL363585

Cc1ccccc1C(C/C(=N\O)c1c[nH]c(=O)c(C)c1)c1ccc(C(=O)NCCCC(=O)O)cc1

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 4/20 0.45
BRD4 O60885 1/20 0.39
EPHX2 P34913 1/20 0.38
MAPK1 P28482 1/20 0.37
NR1H4 Q96RI1 2/20 0.36
MAPK8 P45983 1/20 0.36
PPARA Q07869 1/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
PPARG P37231 1/20 0.36
FOLH1 Q04609 1/20 0.36
GCG P01275 4/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL364071 0.95 GPBAR1 (0.47) GPBAR1BRD4EPHX2GCG
SCHEMBL363667 0.91 GPBAR1 (0.42) GPBAR1BRD4EPHX2SMN1; SMN2
SCHEMBL364032 0.91 GPBAR1 (0.47) GPBAR1BRD4EPHX2MAPK1NPC1
SCHEMBL362350 0.90 GPBAR1 (0.48) GPBAR1BRD4EPHX2SMN1; SMN2
SCHEMBL363032 0.87 GPBAR1 (0.45) GPBAR1BRD4EPHX2
SCHEMBL363542 0.86 GPBAR1 (0.47) GPBAR1BRD4EPHX2MAPK1NPC1
SCHEMBL364239 0.86 GPBAR1 (0.47) GPBAR1BRD4EPHX2MAPK1NPC1
SCHEMBL362902 0.85 GPBAR1 (0.45) GPBAR1BRD4EPHX2MAPK1
SCHEMBL363678 0.85 GPBAR1 (0.61) GPBAR1BRD4
SCHEMBL364242 0.83 GPBAR1 (0.44) GPBAR1BRD4EPHX2MAPK1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP claimed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO claimed
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed