SCHEMBL362350

SCHEMBL362350

Cc1ccccc1C(C/C(=N\O)c1c[nH]c(=O)c(C)c1)c1ccc(C(=O)NCC(=O)O)cc1

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 4/20 0.48
BRD4 O60885 1/20 0.41
SLC6A9 P48067 2/20 0.40
PTPRC P08575 2/20 0.38
CTSL P07711 1/20 0.38
PTPN13 Q12923 1/20 0.38
TYMS P04818 1/20 0.37
EPHX2 P34913 1/20 0.36
CTSA P10619 4/20 0.35
USP5 P45974 1/20 0.35
GART P22102 1/20 0.34
KDM4E B2RXH2 1/20 0.33
MAPT P10636 1/20 0.33
HIF1A Q16665 1/20 0.33
SLC22A6 Q4U2R8 1/20 0.33
SLC22A8 Q8TCC7 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP3A4 P08684 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL364071 0.91 GPBAR1 (0.47) GPBAR1BRD4EPHX2
SCHEMBL364032 0.90 GPBAR1 (0.47) GPBAR1BRD4SLC6A9EPHX2KDM4E
SCHEMBL363585 0.90 GPBAR1 (0.45) GPBAR1BRD4EPHX2SMN1; SMN2
SCHEMBL364239 0.89 GPBAR1 (0.47) GPBAR1BRD4SLC6A9EPHX2KDM4E
SCHEMBL363542 0.89 GPBAR1 (0.47) GPBAR1BRD4SLC6A9EPHX2KDM4E
SCHEMBL362902 0.88 GPBAR1 (0.45) GPBAR1BRD4SLC6A9EPHX2KDM4E
SCHEMBL363678 0.88 GPBAR1 (0.61) GPBAR1BRD4CTSACYP3A4
SCHEMBL363032 0.87 GPBAR1 (0.45) GPBAR1BRD4SLC6A9EPHX2
SCHEMBL363289 0.86 GPBAR1 (0.41) GPBAR1BRD4SLC6A9EPHX2KDM4E
SCHEMBL364242 0.86 GPBAR1 (0.44) GPBAR1BRD4SLC6A9EPHX2CTSA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP claimed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO claimed
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed