SCHEMBL365274

SCHEMBL365274

Cc1cc(Cl)ccc1C(C/C(=N\O)c1c[nH]c(=O)c(C)c1)c1ccc(C(=O)O)cc1

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 4/20 0.46
BRD4 O60885 1/20 0.35
SPR P35270 1/20 0.34
MGAM O43451 2/20 0.34
GAA P10253 2/20 0.34
SI P14410 2/20 0.34
MGAM2 Q2M2H8 2/20 0.34
GRM1 Q13255 2/20 0.34
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
CYP1A2 P05177 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
POLB P06746 2/20 0.33
KEAP1 Q14145 1/20 0.33
NFE2L2 Q16236 1/20 0.33
PRKCZ Q05513 1/20 0.32
RXRA P19793 1/20 0.31
SLC6A3 Q01959 1/20 0.31
MRGPRX4 Q96LA9 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL363178 0.97 GPBAR1 (0.51) GPBAR1BRD4SPRMGAMGAA
SCHEMBL361680 0.89 GPBAR1 (0.47) GPBAR1BRD4SPRMGAMGAA
SCHEMBL12505651 0.88 GPBAR1 (0.35) GPBAR1BRD4MGAMGAASI
SCHEMBL364331 0.88 MGAM (0.43) GPBAR1BRD4SPRMGAMGAA
SCHEMBL362795 0.88 GPBAR1 (0.36) GPBAR1BRD4MEN1KMT2APOLB
SCHEMBL365756 0.87 ADRB3 (0.38) GPBAR1MEN1KMT2APOLBMRGPRX4
SCHEMBL363678 0.87 GPBAR1 (0.61) GPBAR1BRD4MGAMGAASI
SCHEMBL365294 0.87 GPBAR1 (0.35) GPBAR1BRD4GAAMEN1KMT2A
SCHEMBL363289 0.86 GPBAR1 (0.41) GPBAR1BRD4MEN1KMT2ACYP1A2
SCHEMBL363235 0.86 GPBAR1 (0.51) GPBAR1BRD4GRM1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP claimed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO claimed
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed