SCHEMBL3637441

SCHEMBL3637441

COc1cc(Nc2nc(CC(C)c3cc(F)c(F)c(F)c3)cs2)ccc1-c1nc(C)c[nH]1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLA2G7 Q13093 3/20 0.39
MAPT P10636 4/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
GAA P10253 2/20 0.34
NPC1 O15118 2/20 0.34
ALDH1A1 P00352 2/20 0.34
RAB9A P51151 2/20 0.34
NFKB1 P19838 1/20 0.34
NFKB2 Q00653 1/20 0.34
RELA Q04206 1/20 0.34
IMPDH2 P12268 1/20 0.34
CYP1B1 Q16678 3/20 0.34
CYP1A1 P04798 2/20 0.34
ALOX5 P09917 1/20 0.34
PTGES O14684 1/20 0.34
CYP1A2 P05177 1/20 0.34
PSEN1 P49768 3/20 0.34
PSEN2 P49810 3/20 0.34
APH1B Q8WW43 3/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3636479 0.86 IMPDH2 (0.35) PLA2G7MAPTMEN1KMT2AIMPDH2
SCHEMBL3640999 0.80 CYP1B1 (0.53) MAPTMEN1KMT2AGAANPC1
SCHEMBL3634963 0.79 MAPT (0.40) PLA2G7MAPTMEN1KMT2AGAA
Hydrochloric Acid SCHEMBL3635538 0.79 PLA2G7 (0.37) PLA2G7MAPTMEN1KMT2AGAA
SCHEMBL3638760 0.79 PSEN1 (0.48) MAPTMEN1KMT2AGAAALDH1A1
SCHEMBL1040135 0.78 MAPT (0.46) MAPTMEN1KMT2AGAAALDH1A1
SCHEMBL3633741 0.78 PLA2G7 (0.37) PLA2G7MAPTMEN1KMT2AGAA
SCHEMBL3636568 0.78 PLA2G7 (0.34) PLA2G7MAPTMEN1KMT2ARAB9A
SCHEMBL3633324 0.78 CCNT1 (0.41) PLA2G7MAPTMEN1KMT2ANPC1
SCHEMBL3637440 0.77 TP53 (0.40) PLA2G7MAPTMEN1KMT2AGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2155740-A1 HETARYLANILINES AS MODULATORS FOR AMYLOID BETA F. Hoffmann-Roche AG (CH) 2010-02-24 EP disclosed
WO-2008138753-A1 HETARYLANILINES AS MODULATORS FOR AMYLOID BETA F. HOFFMANN-LA ROCHE AG (CH) 2008-11-20 WO disclosed