SCHEMBL3638899

SCHEMBL3638899

COc1cc(Nc2ncc(CNc3ccc(F)cc3)s2)ccc1-c1nc(C)c[nH]1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIT P10721 3/20 0.39
PLK1 P53350 1/20 0.38
KCNH2 Q12809 1/20 0.38
GPX4 P36969 3/20 0.37
GRIN1 Q05586 2/20 0.35
GRIN2B Q13224 2/20 0.35
CLK1 P49759 1/20 0.35
DYRK1A Q13627 1/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
GPR55 Q9Y2T6 2/20 0.35
EGFR P00533 1/20 0.35
ERBB2 P04626 1/20 0.35
IGF1R P08069 1/20 0.35
TEK Q02763 1/20 0.35
MAP3K11 Q16584 2/20 0.34
AAK1 Q2M2I8 1/20 0.34
PSEN1 P49768 1/20 0.34
PSEN2 P49810 1/20 0.34
APH1B Q8WW43 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3633316 0.84 PIK3CD (0.34) KITGPX4GRIN1GRIN2BEGFR
SCHEMBL3634899 0.82 LMNA (0.44) EGFRERBB2IGF1RTEKPSEN1
SCHEMBL3635336 0.82 KCNH2 (0.42) KCNH2GRIN2BMEN1KMT2APSEN1
SCHEMBL3638040 0.80 OGA (0.44) GPX4PSEN1PSEN2APH1BNCSTN
SCHEMBL3636918 0.79 MAP4K1 (0.44) KITCDK9
SCHEMBL3638880 0.78 PSEN1 (0.38) KITPLK1GPX4EGFRERBB2
SCHEMBL1040502 0.78 PSEN1 (0.56) KCNH2PSEN1PSEN2APH1BNCSTN
SCHEMBL3406352 0.75 BRAF (0.46) KCNH2EGFRPSEN1PSEN2APH1B
SCHEMBL3640777 0.74 PSEN1 (0.52) KITPLK1MEN1KMT2AEGFR
SCHEMBL2329626 0.73 MAPT (0.45) KCNH2GRIN2BKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2155740-A1 HETARYLANILINES AS MODULATORS FOR AMYLOID BETA F. Hoffmann-Roche AG (CH) 2010-02-24 EP disclosed
WO-2008138753-A1 HETARYLANILINES AS MODULATORS FOR AMYLOID BETA F. HOFFMANN-LA ROCHE AG (CH) 2008-11-20 WO disclosed