SCHEMBL3639612

SCHEMBL3639612

Fc1c(C(Br)Br)ccc(Cl)c1Oc1cc(Cl)cc(Br)c1

nearest known ligand 0.31

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
EPAS1 Q99814 4/20 0.31
CYP3A4 P08684 1/20 0.31
VEGFA P15692 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3031283 0.80 EPAS1 (0.33) EPAS1CYP3A4
SCHEMBL14920185 0.78 RHEB (0.45)
SCHEMBL3023318 0.78 CYP3A4 (0.38) EPAS1CYP3A4
SCHEMBL13481896 0.77 CYP3A4 (0.42) EPAS1CYP3A4
SCHEMBL3033047 0.77 CYP3A4 (0.38) EPAS1CYP3A4
SCHEMBL4754754 0.73 CAMK2A (0.41) CYP3A4
SCHEMBL2884075 0.72 EPAS1 (0.40) EPAS1VEGFA
SCHEMBL13581458 0.72 CYP3A4 (0.34) CYP3A4
SCHEMBL2884469 0.71 TSHR (0.32) CYP3A4
SCHEMBL4752685 0.70 MEP1B (0.38) CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2166856-A1 CHEMICAL COMPOUNDS GlaxoSmithKline LLC (US) 2010-03-31 EP disclosed
WO-2008154271-A1 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2008-12-18 WO disclosed