SCHEMBL4754754

SCHEMBL4754754

O=C(O)Cc1ccc(Cl)c(Oc2cc(Cl)cc(Br)c2)c1F

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CAMK2A Q9UQM7 3/20 0.41
THRA P10827 7/20 0.39
THRB P10828 7/20 0.39
CYP3A4 P08684 2/20 0.38
CHRM1 P11229 1/20 0.36
MEP1B Q16820 1/20 0.36
CXCL8 P10145 2/20 0.35
GRIK1 P39086 1/20 0.34
CYP2C9 P11712 2/20 0.34
CYP2C19 P33261 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4754909 0.88 THRA (0.36) CAMK2ATHRATHRBCYP3A4CHRM1
SCHEMBL4752685 0.86 MEP1B (0.38) CYP3A4MEP1BCYP2C9CYP2C19
SCHEMBL16175471 0.85 CYP3A4 (0.46) CAMK2ATHRATHRBCYP3A4CHRM1
SCHEMBL2340437 0.85 CYP3A4 (0.37) THRBCYP3A4MEP1BCYP2C9CYP2C19
SCHEMBL13481896 0.85 CYP3A4 (0.42) CYP3A4MEP1BCYP2C9CYP2C19
SCHEMBL3038920 0.84 CYP1A2 (0.41) CAMK2ATHRATHRBGRIK1
SCHEMBL4752770 0.84 CYP1A2 (0.41) CAMK2ATHRATHRBGRIK1
SCHEMBL3023318 0.83 CYP3A4 (0.38) CYP3A4MEP1BCYP2C9CYP2C19
SCHEMBL1344613 0.82 CYP3A4 (0.55) CAMK2ATHRATHRBCYP3A4CHRM1
SCHEMBL13236609 0.82 CAMK2A (0.39) CAMK2ATHRATHRBCYP3A4CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008157273-A1 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2008-12-24 WO disclosed
WO-2008157330-A1 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2008-12-24 WO disclosed