SCHEMBL4752685

SCHEMBL4752685

NNC(=O)Cc1ccc(Cl)c(Oc2cc(Cl)cc(Br)c2)c1F

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MEP1B Q16820 2/20 0.38
ALDH1A1 P00352 3/20 0.36
MAPT P10636 1/20 0.36
CYP3A4 P08684 2/20 0.35
POLB P06746 1/20 0.34
ERCC1 P07992 1/20 0.34
ERCC4 Q92889 1/20 0.34
PLA2G2A P14555 1/20 0.33
TLR8 Q9NR97 1/20 0.32
P2RX7 Q99572 1/20 0.32
TAOK1 Q7L7X3 1/20 0.32
TAOK3 Q9H2K8 1/20 0.32
LMNA P02545 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
CARM1 Q86X55 1/20 0.31
PRMT6 Q96LA8 1/20 0.31
MEP1A Q16819 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4754754 0.86 CAMK2A (0.41) MEP1BCYP3A4CYP2C9CYP2C19
SCHEMBL4754828 0.84 CYP3A4 (0.51) MEP1BALDH1A1MAPTCYP3A4POLB
SCHEMBL2340437 0.81 CYP3A4 (0.37) MEP1BALDH1A1MAPTCYP3A4POLB
SCHEMBL3033047 0.81 CYP3A4 (0.38) MEP1BCYP3A4CYP2C9CYP2C19
SCHEMBL13481896 0.81 CYP3A4 (0.42) MEP1BCYP3A4CYP2C9CYP2C19
SCHEMBL13984460 0.80 TDP1 (0.44) MEP1BALDH1A1MAPTPOLBLMNA
SCHEMBL3023318 0.80 CYP3A4 (0.38) MEP1BCYP3A4CYP2C9CYP2C19
SCHEMBL13984632 0.78 ALDH1A1 (0.46) ALDH1A1MAPTCYP3A4POLBLMNA
SCHEMBL4754790 0.78 CYP3A4 (0.44) ALDH1A1MAPTCYP3A4CYP2C9CYP2C19
SCHEMBL4754909 0.77 THRA (0.36) ALDH1A1MAPTCYP3A4LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008157273-A1 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2008-12-24 WO disclosed
WO-2008157330-A1 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2008-12-24 WO disclosed
WO-2008157330-A1 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2008-12-24 WO disclosed
WO-2008157273-A1 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2008-12-24 WO disclosed