SCHEMBL3640686

SCHEMBL3640686

Cc1ccc([C@@H](C)NC(=O)c2cccc(C(N)=O)c2)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.55
TAS1R3 Q7RTX0 1/20 0.54
TAS1R1 Q7RTX1 1/20 0.54
SMN1; SMN2 Q16637 2/20 0.51
PARP1 P09874 1/20 0.50
LMNA P02545 3/20 0.49
GPR139 Q6DWJ6 1/20 0.48
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
CYP1A2 P05177 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
CA2 P00918 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
MAPK1 P28482 1/20 0.46
F2 P00734 1/20 0.46
F10 P00742 1/20 0.46
PRSS1 P07477 1/20 0.46
PHGDH O43175 2/20 0.46
ANPEP P15144 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3345042 0.88 ALDH1A1 (0.69) ALDH1A1SMN1; SMN2LMNAGPR139MEN1
SCHEMBL3646228 0.88 ALDH1A1 (0.69) ALDH1A1SMN1; SMN2LMNAGPR139MEN1
SCHEMBL3351175 0.88 ALDH1A1 (0.69) ALDH1A1SMN1; SMN2LMNAGPR139MEN1
SCHEMBL9318785 0.82 SMN1; SMN2 (0.73) ALDH1A1TAS1R3TAS1R1SMN1; SMN2LMNA
SCHEMBL28651689 0.82 SMN1; SMN2 (0.73) ALDH1A1TAS1R3TAS1R1SMN1; SMN2LMNA
SCHEMBL2977147 0.80 NPSR1 (0.59) ALDH1A1PARP1KMT2AANPEP
P-Xylene SCHEMBL17907442 0.79 PARP1 (0.76) ALDH1A1PARP1LMNACYP2C19TDP1
SCHEMBL3686677 0.79 ALDH1A1 (0.60) ALDH1A1SMN1; SMN2LMNAMEN1KMT2A
SCHEMBL3648293 0.79 ALDH1A1 (0.47) ALDH1A1SMN1; SMN2PARP1LMNAMEN1
SCHEMBL3643873 0.78 PARP1 (0.44) ALDH1A1TAS1R3TAS1R1PARP1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2178837-A2 ISOPHTHALAMIDE DERIVATIVES INHIBITING BETA-SECRETASE ACTIVITY COMENTIS, INC. (US) 2010-04-28 EP claimed
WO-2009015369-A2 COMPOUNDS WHICH INHIBIT BETA-SECRETASE ACTIVITY AND METHODS OF USE THEREOF COMENTIS, INC. (US) 2009-01-29 WO claimed