SCHEMBL364099

SCHEMBL364099

OC1CNCCC12CCN(c1ccc(CC(F)(F)F)cc1)C2

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 2/20 0.44
SLC6A4 P31645 2/20 0.44
SLC6A3 Q01959 2/20 0.44
LIPE Q05469 4/20 0.38
PANK3 Q9H999 2/20 0.32
ME2 P23368 1/20 0.31
ME1 P48163 1/20 0.31
ME3 Q16798 1/20 0.31
USP2 O75604 3/20 0.30
CYP2D6 P10635 3/20 0.30
ALDH1A1 P00352 2/20 0.30
CYP3A4 P08684 2/20 0.30
TSHR P16473 2/20 0.30
CYP2C19 P33261 2/20 0.30
TP53 P04637 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP2C9 P11712 1/20 0.30
HPGD P15428 1/20 0.30
MAPK1 P28482 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30330141 0.69 ADRB1 (0.52) USP2ALDH1A1TSHRHSD17B10
SCHEMBL17608949 0.67 TSHR (0.52) CYP2D6ALDH1A1CYP3A4TSHRCYP2C19
SCHEMBL11371 0.65 KCNH2 (0.34) LIPEUSP2CYP2D6ALDH1A1CYP3A4
SCHEMBL5578 0.65 LIPE (0.34) LIPEUSP2ALDH1A1CYP3A4TSHR
SCHEMBL746750 0.64 CYP3A4 (0.44) LIPEUSP2CYP2D6ALDH1A1CYP3A4
SCHEMBL16862199 0.64 TSHR (0.58) CYP2D6ALDH1A1CYP3A4TSHRCYP2C19
SCHEMBL19320638 0.63 SLC6A2 (0.34) SLC6A2SLC6A4SLC6A3
SCHEMBL17611694 0.63 OPRM1 (0.43) SLC6A2SLC6A4SLC6A3USP2CYP2D6
SCHEMBL19341570 0.62 USP2 (0.52) USP2CYP2D6ALDH1A1CYP3A4TSHR
SCHEMBL1946683 0.62 LIPE (0.47) LIPE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593454-A1 NEW AZACYCLIC COMPOUNDS F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007367-A1 NEW AZACYCLIC COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed