SCHEMBL364253

SCHEMBL364253

CCc1ccc(OCc2ccc(C(=O)NS(C)(=O)=O)c(F)c2)cc1

nearest known ligand 0.53

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 15/20 0.53
SCN5A Q14524 2/20 0.53
MAOB P27338 4/20 0.47
MAOA P21397 2/20 0.47
RXRA P19793 1/20 0.45
RXRB P28702 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Diethylamine SCHEMBL16239835 0.96 SCN9A (0.49) SCN9ASCN5AMAOBMAOARXRA
SCHEMBL363861 0.87 RXRA (0.49) SCN9ASCN5ARXRARXRB
SCHEMBL366513 0.85 PTGER4 (0.47) SCN9ASCN5ARXRARXRB
Diethylamine SCHEMBL16240278 0.83 RXRA (0.45) SCN9ASCN5ARXRARXRB
Diethylamine SCHEMBL16239544 0.81 ADRB1 (0.44) SCN9ASCN5ARXRARXRB
SCHEMBL364950 0.81 MAOB (0.66) SCN9ASCN5AMAOBMAOA
SCHEMBL364340 0.80 RXRA (0.62) SCN9ARXRARXRB
SCHEMBL365348 0.78 SCN9A (0.56) SCN9ASCN5AMAOBMAOA
Diethylamine SCHEMBL16239678 0.76 RXRA (0.57) SCN9ARXRARXRB
SCHEMBL16240191 0.75 SCN9A (0.76) SCN9ASCN5AMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9096500-B2 Acyl sulfonamide compounds PFIZER LIMITED (GB) 2015-08-04 US disclosed
EP-2593428-A2 N-SULFONYLBENZAMIDES AS INHIBITORS OF VOLTAGE-GATED SODIUM CHANNELS Pfizer Limited (GB) 2013-05-22 EP disclosed
US-20130109701-A1 Chemical Compounds PFIZER LIMITED (GB) 2013-05-02 US disclosed
WO-2012007868-A2 CHEMICAL COMPOUNDS PFIZER LIMITED (GB) 2012-01-19 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130109701-A1 Chemical Compounds SCN1A, SCN1B, SCN7A SCN9A 16/4885SCN5A 5/4885MAOB 3660/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.