SCHEMBL364586

SCHEMBL364586

Cc1ccccc1[C@@](C/C=N/O)(c1ccc(-c2ccc(C(=O)O)cc2)cc1)c1cc(Cl)ncc1F

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 3/20 0.34
EPHX2 P34913 1/20 0.32
MAP4K4 O95819 4/20 0.32
KCNQ3 O43525 2/20 0.32
KCNQ2 O43526 2/20 0.32
RXRA P19793 2/20 0.31
RXRB P28702 2/20 0.31
TRPM8 Q7Z2W7 2/20 0.31
MEN1 O00255 1/20 0.30
NPC1 O15118 1/20 0.30
GAA P10253 1/20 0.30
MAPT P10636 1/20 0.30
RAB9A P51151 1/20 0.30
KMT2A Q03164 1/20 0.30
PDK2 Q15119 1/20 0.30
KCNE1 P15382 1/20 0.30
KCNQ1 P51787 1/20 0.30
LMNA P02545 1/20 0.30
POLB P06746 1/20 0.30
PIN1 Q13526 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL371307 0.86 MAP4K4 (0.34) GPBAR1EPHX2MAP4K4RXRARXRB
SCHEMBL363808 0.85
SCHEMBL364476 0.80 NFE2L2 (0.33)
SCHEMBL370899 0.80 GPBAR1 (0.38) GPBAR1EPHX2RXRARXRBLMNA
SCHEMBL370897 0.80 GPBAR1 (0.38) GPBAR1EPHX2RXRARXRBLMNA
SCHEMBL364577 0.70 CYP19A1 (0.32)
SCHEMBL361805 0.69
SCHEMBL362947 0.68
SCHEMBL362408 0.68 NFE2L2 (0.35)
SCHEMBL363380 0.67 KIF11 (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed