SCHEMBL370897

SCHEMBL370897

Cc1cc([C@@](C/C=N/O)(c2ccc(-c3ccc(C(=O)O)cc3)cc2)c2ccccc2C)cc(C)n1

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 2/20 0.38
NR1H4 Q96RI1 1/20 0.35
VCP P55072 3/20 0.35
RXRA P19793 6/20 0.34
RXRB P28702 5/20 0.34
EPHX2 P34913 1/20 0.34
EDNRB P24530 1/20 0.34
EDNRA P25101 1/20 0.34
RXRG P48443 1/20 0.34
LMNA P02545 1/20 0.34
POLB P06746 1/20 0.34
PTGES O14684 1/20 0.32
ALOX5 P09917 1/20 0.32
GRM5 P41594 1/20 0.32
RARA P10276 1/20 0.32
RARB P10826 1/20 0.32
RARG P13631 1/20 0.32
BCL2 P10415 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL364586 0.80 GPBAR1 (0.34) GPBAR1RXRARXRBEPHX2LMNA
SCHEMBL364577 0.73 CYP19A1 (0.32)
SCHEMBL362336 0.72 KIF11 (0.32)
SCHEMBL362349 0.71 TTR (0.31) ALOX5
SCHEMBL364014 0.70
SCHEMBL362881 0.69 CHRM3 (0.37) EDNRBEDNRA
SCHEMBL8119878 0.66 RXRA (0.66) RXRARXRBRXRGPOLB
SCHEMBL370900 0.62 GPBAR1 (0.80) GPBAR1NR1H4VCPRXRARXRB
SCHEMBL1390281 0.62 GPBAR1 (0.80) GPBAR1NR1H4VCPRXRARXRB
SCHEMBL364364 0.61 GPBAR1 (0.63) GPBAR1NR1H4VCPRXRARXRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed