SCHEMBL3645987

SCHEMBL3645987

CN(Cc1cc(S(=O)(=O)c2cccnc2)c(-c2cccnc2Cl)s1)C(=O)OC(C)(C)C

nearest known ligand 0.36

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 1/20 0.36
RXFP1 Q9HBX9 1/20 0.33
PTGER2 P43116 6/20 0.33
F2 P00734 2/20 0.32
NAMPT P43490 2/20 0.32
HTR2C P28335 1/20 0.32
SLC6A4 P31645 1/20 0.32
ABCC9 O60706 1/20 0.31
ABCC8 Q09428 1/20 0.31
KCNJ11 Q14654 1/20 0.31
KCNJ8 Q15842 1/20 0.31
POLB P06746 2/20 0.31
CLK1 P49759 1/20 0.31
GLS O94925 1/20 0.31
SOS1 Q07889 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3653190 0.91 ABCC9 (0.33) GPBAR1PTGER2F2NAMPTABCC9
SCHEMBL4126083 0.89 GPBAR1 (0.36) GPBAR1RXFP1PTGER2NAMPTPOLB
SCHEMBL3648432 0.88 GPBAR1 (0.39) GPBAR1RXFP1PTGER2F2NAMPT
SCHEMBL3654491 0.87 NAMPT (0.35) GPBAR1PTGER2F2NAMPTABCC9
SCHEMBL3645990 0.82 PTGER2 (0.35) GPBAR1RXFP1PTGER2NAMPTABCC9
SCHEMBL3649650 0.82 NAMPT (0.36) PTGER2F2NAMPTHTR2CSLC6A4
SCHEMBL3650554 0.80 HTR2C (0.37) GPBAR1RXFP1F2NAMPTHTR2C
SCHEMBL4126584 0.79 NAMPT (0.37) GPBAR1PTGER2NAMPTABCC9ABCC8
Fumaric Acid SCHEMBL3650347 0.78 TBXAS1 (0.36) NAMPTPOLB
Fumaric Acid SCHEMBL3650341 0.78 TBXAS1 (0.36) NAMPTPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2190822-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2010-06-02 EP disclosed
WO-2009041705-A9 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL (JP) 2009-08-13 WO disclosed
WO-2009041705-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-04-02 WO disclosed