SCHEMBL364613

SCHEMBL364613

O=C(O)Oc1ccc(-c2cccnc2)o1

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 13/20 0.51
CYP3A4 P08684 9/20 0.51
CYP2C19 P33261 8/20 0.51
CYP2D6 P10635 7/20 0.51
CYP2C9 P11712 7/20 0.51
CYP2E1 P05181 6/20 0.51
CYP2B6 P20813 6/20 0.51
MKNK1 Q9BUB5 1/20 0.44
MKNK2 Q9HBH9 1/20 0.44
ALDH1A1 P00352 3/20 0.43
CYP1A2 P05177 2/20 0.43
MAPT P10636 1/20 0.43
MAPK1 P28482 1/20 0.43
KDM4E B2RXH2 1/20 0.42
NPC1 O15118 1/20 0.42
HPGD P15428 1/20 0.42
RAB9A P51151 1/20 0.42
HSD17B10 Q99714 1/20 0.42
KMO O15229 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2724814 0.78 ALDH1A1 (0.51) CYP2A6CYP3A4CYP2C19CYP2D6CYP2C9
SCHEMBL370030 0.78 ALDH1A1 (0.55) CYP2A6CYP3A4CYP2C19MKNK1MKNK2
SCHEMBL364612 0.76 ALDH1A1 (0.62) CYP2A6CYP3A4CYP2C19CYP2D6CYP2C9
SCHEMBL23091171 0.75 ALDH1A1 (0.50) CYP2A6CYP3A4CYP2C19CYP2D6CYP2C9
SCHEMBL370075 0.75 CYP2A6 (0.51) CYP2A6CYP3A4CYP2C19CYP2C9CYP2E1
SCHEMBL21249436 0.75 ALDH1A1 (0.62) CYP2A6CYP3A4CYP2C19CYP2D6CYP2C9
SCHEMBL27605095 0.74 CYP2A6 (0.57) CYP2A6CYP3A4CYP2C19CYP2D6CYP2C9
SCHEMBL369291 0.74 SCD (0.49) CYP3A4CYP2C19CYP2D6CYP2C9MKNK1
SCHEMBL23091243 0.74 KMT2A (0.52) CYP2A6CYP3A4CYP2C19CYP2D6CYP2C9
SCHEMBL363027 0.74 KMO (0.43) CYP2A6CYP3A4CYP2C19CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593447-B1 3-PYRIDYL-HETEROARYLCARBOXAMIDE COMPOUNDS AS PESTICIDES BAYER IP GMBH (DE) 2016-08-17 EP disclosed
EP-2630133-A1 NOVEL HETEROCYCLIC COMPOUNDS AS PESTICIDES Bayer Intellectual Property GmbH (DE) 2013-08-28 EP disclosed
EP-2593447-A2 NEW HETEROCYCLIC COMPOUNDS AS PESTICIDES Bayer Intellectual Property GmbH (DE) 2013-05-22 EP disclosed
WO-2012052412-A1 NOVEL HETEROCYCLIC COMPOUNDS AS PESTICIDES BAYER CROPSCIENCE AG (DE) 2012-04-26 WO disclosed
WO-2012007500-A2 NEW HETEROCYCLIC COMPOUNDS AS PESTICIDES BAYER CROPSCIENCE AG (DE) 2012-01-19 WO disclosed