SCHEMBL3650221

SCHEMBL3650221

CC(C)(C)CN(Cc1nc(-c2cccnc2F)c(Sc2cccc(Cl)c2)s1)C(=O)O

nearest known ligand 0.35

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 1/20 0.35
POLB P06746 2/20 0.33
USP7 Q93009 1/20 0.33
SLC6A9 P48067 3/20 0.33
KDM4E B2RXH2 2/20 0.32
MEN1 O00255 2/20 0.32
HPGD P15428 2/20 0.32
KMT2A Q03164 2/20 0.32
ALDH1A1 P00352 1/20 0.32
PKM P14618 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
GAA P10253 1/20 0.31
MAPT P10636 1/20 0.31
MAPK14 Q16539 1/20 0.31
TP53 P04637 1/20 0.31
RXFP1 Q9HBX9 1/20 0.31
ROCK2 O75116 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3655562 0.90 DHODH (0.33) DHODH
SCHEMBL3653706 0.90 DHODH (0.32) DHODHROCK2
SCHEMBL4118235 0.87 DHODH (0.37) DHODHPOLBUSP7SLC6A9KDM4E
SCHEMBL3650214 0.83 SLC6A9 (0.34) DHODHPOLBUSP7SLC6A9KDM4E
SCHEMBL3646797 0.81 HSD11B1 (0.35) DHODH
SCHEMBL3650216 0.80 POLB (0.36) DHODHPOLBUSP7SLC6A9KDM4E
SCHEMBL3650619 0.80 ALDH1A1 (0.32) POLBHPGDALDH1A1L3MBTL1GAA
SCHEMBL4118238 0.79 POLB (0.39) DHODHPOLBUSP7SLC6A9KDM4E
SCHEMBL3647079 0.78
SCHEMBL3652263 0.78 DHODH (0.34) DHODHPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2190822-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2010-06-02 EP disclosed
WO-2009041705-A9 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL (JP) 2009-08-13 WO disclosed
WO-2009041705-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-04-02 WO disclosed