SCHEMBL3655385

SCHEMBL3655385

Cc1cc(Nc2ccc(NC(=O)c3ccc(Nc4ccnc5ccccc45)cc3)cc2)nc(N)n1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DNMT1 P26358 13/20 1.00
DNMT3A Q9Y6K1 9/20 1.00
DNMT3L Q9UJW3 6/20 1.00
EHMT1 Q9H9B1 3/20 1.00
MYC P01106 1/20 1.00
MAP2K3 P46734 1/20 1.00
EHMT2 Q96KQ7 1/20 1.00
DNMT3B Q9UBC3 1/20 1.00
HDAC3 O15379 1/20 0.57
ACHE P22303 1/20 0.57
HDAC1 Q13547 1/20 0.57
HDAC7 Q8WUI4 1/20 0.57
HDAC2 Q92769 1/20 0.57
HDAC8 Q9BY41 1/20 0.57
HDAC6 Q9UBN7 1/20 0.57
HDAC9 Q9UKV0 1/20 0.57
HDAC5 Q9UQL6 1/20 0.57
AURKA O14965 1/20 0.48
AURKB Q96GD4 1/20 0.48
MAPT P10636 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3786360 1.00 DNMT1 (1.00) DNMT1DNMT3ADNMT3LEHMT1MYC
SCHEMBL29351315 1.00 DNMT1 (1.00) DNMT1DNMT3ADNMT3LEHMT1MYC
Hydrochloric Acid SCHEMBL1886043 0.99 DNMT1 (0.98) DNMT1DNMT3ADNMT3LEHMT1MYC
Hydrochloric Acid SCHEMBL1880676 0.99 DNMT1 (0.98) DNMT1DNMT3ADNMT3LEHMT1MYC
SCHEMBL3657042 0.94 DNMT1 (1.00) DNMT1DNMT3ADNMT3LEHMT1MYC
Hydrochloric Acid SCHEMBL1880578 0.94 DNMT1 (0.98) DNMT1DNMT3ADNMT3LEHMT1MYC
SCHEMBL3789536 0.93 DNMT1 (1.00) DNMT1DNMT3ADNMT3LEHMT1MYC
SCHEMBL3800388 0.92 DNMT1 (0.85) DNMT1DNMT3ADNMT3LEHMT1MYC
SCHEMBL3784380 0.92 DNMT1 (0.85) DNMT1DNMT3ADNMT3LEHMT1MYC
Hydrochloric Acid SCHEMBL1878590 0.92 DNMT1 (0.98) DNMT1DNMT3ADNMT3LEHMT1MYC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 47 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11992500-B2 Use of methylation inhibitors for the treatment of autoimmune diseases RUSH UNIVERSITY MEDICAL CENTER (US) 2024-05-28 US claimed
US-20210128600-A1 Use of Methylation Inhibitors for the Treatment of Autoimmune Diseases RUSH UNIVERSITY MEDICAL CENTER (US) 2021-05-06 US claimed
EP-3207932-A1 DNA METHYLTRANSFERASE INHIBITORS FOR RETT SYNDROME THERAPY Universität Stuttgart (DE) 2017-08-23 EP claimed
US-20250295686-A1 COMBINATION DECITABINE AND MPS1 INHIBITOR THERAPY TO PRIME CANCER IMMUNOGENICITY DANA-FARBER CANCER INSTITUTE, INC. 2025-09-25 US disclosed
US-11992500-B2 Use of methylation inhibitors for the treatment of autoimmune diseases RUSH UNIVERSITY MEDICAL CENTER (US) 2024-05-28 US disclosed
US-20240125787-A1 STING LEVELS AS A BIOMARKER FOR CANCER IMMUNOTHERAPY DANA-FARBER CANCER INSTITUTE, INC. (US) 2024-04-18 US disclosed
US-11874276-B2 STING levels as a biomarker for cancer immunotherapy DANA-FARBER CANCER INSTITUTE, INC. (US) 2024-01-16 US disclosed
US-20230346879-A1 COMPOSITIONS AND METHODS FOR COMBINATORIAL DRUG DISCOVERY IN NANOLITER DROPLETS MASSACHUSETTS INSTITUTE OF TECHNOLOGY 2023-11-02 US disclosed
WO-2023069943-A1 COMBINATION DECITABINE AND MPS1 INHIBITOR THERAPY TO PRIME CANCER IMMUNOGENICITY DANA-FARBER CANCER INSTITUTE, INC. (US) 2023-04-27 WO disclosed
US-11564970-B2 Compositions and methods for combinatorial drug discovery in nanoliter droplets THE BROAD INSTITUTE, INC. (US) 2023-01-31 US disclosed
US-11092602-B2 Methods and compositions relating to proteasome inhibitor resistance WHITEHEAD INSTITUTE FOR BIOMEDICAL RESEARCH (US) 2021-08-17 US disclosed
EP-2078008-A2 QUINOLINE DERIVATIVES FOR MODULATING DNA METHYLATION SuperGen, Inc. (US) 2009-07-15 EP disclosed
US-20090099106-A1 QUINOLINE DERIVATIVES FOR MODULATING DNA METHYLATION SUPERGEN, INC. (US) 2009-04-16 US disclosed
US-20090099106-A1 QUINOLINE DERIVATIVES FOR MODULATING DNA METHYLATION SUPERGEN, INC. (US) 2009-04-16 US disclosed
US-20090099106-A1 QUINOLINE DERIVATIVES FOR MODULATING DNA METHYLATION SUPERGEN, INC. (US) 2009-04-16 US disclosed
WO-2009049132-A1 QUINOLINE DERIVATIVES FOR MODULATING DNA METHYLATION SUPERGEN, INC. (US) 2009-04-16 WO disclosed
WO-2009049132-A1 QUINOLINE DERIVATIVES FOR MODULATING DNA METHYLATION SUPERGEN, INC. (US) 2009-04-16 WO disclosed
US-20080175814-A1 QUINOLINE DERIVATIVES FOR MODULATING DNA METHYLATION SUPERGEN, INC. (US) 2008-07-24 US disclosed
US-20080175814-A1 QUINOLINE DERIVATIVES FOR MODULATING DNA METHYLATION SUPERGEN, INC. (US) 2008-07-24 US disclosed
WO-2008046085-A2 QUINOLINE DERIVATIVES FOR MODULATING DNA METHYLATION SUPERGEN, INC. (US) 2008-04-17 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230346879-A1 COMPOSITIONS AND METHODS FOR COMBINATORIAL DRUG DISCOVERY IN NANOLITER DROPLETS RAB5IF, CLTB, TBK1 DNMT1 4323/4885DNMT3A 3754/4885DNMT3L 4078/4885
US-20080175814-A1 QUINOLINE DERIVATIVES FOR MODULATING DNA METHYLATION DNMT1, DNMT3A, DNMT3L DNMT1 1/4885DNMT3A 2/4885DNMT3L 3/4885
US-11092602-B2 Methods and compositions relating to proteasome inhibitor resistance PSMG3, PSMB1, PSMB11 DNMT1 2760/4885DNMT3A 3574/4885DNMT3L 2739/4885
US-20090099106-A1 QUINOLINE DERIVATIVES FOR MODULATING DNA METHYLATION DNMT1, DNMT3A, DNMT3L DNMT1 1/4885DNMT3A 2/4885DNMT3L 3/4885
US-11564970-B2 Compositions and methods for combinatorial drug discovery in nanoliter droplets RAB5IF, LIPA, CLTB DNMT1 4398/4885DNMT3A 3959/4885DNMT3L 4092/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.