SCHEMBL3655641

SCHEMBL3655641

Cc1cc(NC(=O)c2cccc(N(C)C)c2)ccc1[N+]1(C2CCNC2)CCCC1C

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 10/20 0.44
KDM4E B2RXH2 4/20 0.44
MAPT P10636 4/20 0.44
HSD17B10 Q99714 3/20 0.44
ALDH1A1 P00352 3/20 0.44
HPGD P15428 3/20 0.44
BRAF P15056 2/20 0.44
ALOX15 P16050 2/20 0.44
RAF1 P04049 1/20 0.44
TP53 P04637 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C9 P11712 1/20 0.44
MAPK11 Q15759 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
SMO Q99835 1/20 0.43
RAB9A P51151 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
NPC1 O15118 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3656630 0.91 KCNK3 (0.40) KDM4EMAPTHSD17B10ALDH1A1TP53
SCHEMBL3650124 0.86 HSP90AA1 (0.50) KDM4EMAPTALDH1A1HPGDTP53
SCHEMBL3657580 0.86 ESR1 (0.46) MAPK14MAPTBRAFRAF1RAB9A
SCHEMBL3658339 0.84 RAB9A (0.52) KDM4EMAPTALDH1A1TP53TDP1
Trifluoroacetic Acid SCHEMBL3652245 0.84 NPC1 (0.39) KDM4EMAPTTP53RAB9ASMN1; SMN2
SCHEMBL3655153 0.82 NPC1 (0.43) MAPK14KDM4EMAPTALDH1A1ALOX15
SCHEMBL3652477 0.82 ESR1 (0.45) MAPK14RAB9ANPC1
Trifluoroacetic Acid SCHEMBL3657556 0.82 HSP90AA1 (0.45) KDM4EMAPTALDH1A1TP53RAB9A
Trifluoroacetic Acid SCHEMBL3656228 0.80 RAB9A (0.46) MAPTALDH1A1BRAFTP53TDP1
Trifluoroacetic Acid SCHEMBL3650438 0.78

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2212282-A1 SUBSTITUTED N-PHENYL-BIPYRROLIDINE CARBOXAMIDES AND THERAPEUTIC USE THEREOF Sanofi-Aventis (FR) 2010-08-04 EP disclosed
WO-2009052065-A1 SUBSTITUTED N-PHENYL-BIPYRROLIDINE CARBOXAMIDES AND THERAPEUTIC USE THEREOF SANOFI-AVENTIS (FR) 2009-04-23 WO disclosed