SCHEMBL3655153

SCHEMBL3655153

COc1ccc(C(=O)Nc2ccc([N+]3(C4CCNC4)CCCC3C)c(C)c2)cc1

nearest known ligand 0.55

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 7/20 0.43
RAB9A P51151 7/20 0.43
TP53 P04637 5/20 0.43
SMN1; SMN2 Q16637 4/20 0.43
ALOX15 P16050 1/20 0.43
ALDH1A1 P00352 2/20 0.43
MAPT P10636 2/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
KDM4E B2RXH2 1/20 0.42
HTT P42858 1/20 0.42
MAPK14 Q16539 1/20 0.42
NFKB1 P19838 2/20 0.42
NFKB2 Q00653 2/20 0.42
RELA Q04206 2/20 0.42
PKM P14618 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3650124 0.91 HSP90AA1 (0.50) NPC1RAB9ATP53SMN1; SMN2ALDH1A1
SCHEMBL3656630 0.88 KCNK3 (0.40) TP53ALDH1A1MAPTKDM4E
SCHEMBL3652477 0.88 ESR1 (0.45) NPC1RAB9AMEN1KMT2AMAPK14
SCHEMBL3657680 0.87 RAB9A (0.51) NPC1RAB9ATP53SMN1; SMN2ALOX15
Trifluoroacetic Acid SCHEMBL3657556 0.86 HSP90AA1 (0.45) NPC1RAB9ATP53SMN1; SMN2ALDH1A1
Trifluoroacetic Acid SCHEMBL3650438 0.85
SCHEMBL3658339 0.84 RAB9A (0.52) NPC1RAB9ATP53SMN1; SMN2ALDH1A1
Trifluoroacetic Acid SCHEMBL3656237 0.83 MLYCD (0.41) NPC1RAB9AMEN1KMT2A
SCHEMBL3655641 0.82 MAPK14 (0.44) NPC1RAB9ATP53SMN1; SMN2ALOX15
SCHEMBL3657580 0.82 ESR1 (0.46) RAB9AMAPTMEN1KMT2AHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2212282-A1 SUBSTITUTED N-PHENYL-BIPYRROLIDINE CARBOXAMIDES AND THERAPEUTIC USE THEREOF Sanofi-Aventis (FR) 2010-08-04 EP disclosed
WO-2009052065-A1 SUBSTITUTED N-PHENYL-BIPYRROLIDINE CARBOXAMIDES AND THERAPEUTIC USE THEREOF SANOFI-AVENTIS (FR) 2009-04-23 WO disclosed