SCHEMBL3656229

SCHEMBL3656229

COC(=O)c1cc(CC(c2ccc(F)cc2Cl)C(O)C(F)(F)F)ccn1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.38
MRGPRX4 Q96LA9 1/20 0.37
CTSA P10619 1/20 0.37
L3MBTL1 Q9Y468 2/20 0.36
ALOX15 P16050 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
HSD17B10 Q99714 1/20 0.36
MDM2 Q00987 2/20 0.36
MDM4 O15151 1/20 0.36
ACACB O00763 1/20 0.35
PARP1 P09874 1/20 0.35
MAPT P10636 1/20 0.35
NR3C2 P08235 3/20 0.34
NOTUM Q6P988 1/20 0.34
AR P10275 1/20 0.34
ANO1 Q5XXA6 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
CDC7 O00311 1/20 0.33
DBF4 Q9UBU7 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3657207 0.88 MRGPRX4 (0.43) ALDH1A1MRGPRX4CTSAL3MBTL1ALOX15
SCHEMBL3659044 0.85 MRGPRX4 (0.38) MRGPRX4MDM2MDM4
SCHEMBL3653818 0.77 CDC7 (0.38) ALDH1A1MRGPRX4L3MBTL1HSD17B10MAPT
SCHEMBL3658244 0.77 CDC7 (0.37) ALDH1A1MRGPRX4L3MBTL1NPSR1HSD17B10
SCHEMBL3651279 0.76 KMO (0.39) MRGPRX4
SCHEMBL3656161 0.76 P4HTM (0.40) ALDH1A1L3MBTL1ALOX15MDM2MAPT
SCHEMBL3657608 0.76 EIF4E (0.36)
SCHEMBL3659717 0.75 MAPT (0.34) ALDH1A1MAPTMEN1KMT2A
SCHEMBL3659842 0.75 KMO (0.36) MRGPRX4MDM2
SCHEMBL838921 0.73 ALDH1A1 (0.40) ALDH1A1L3MBTL1ALOX15NPSR1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2205562-A1 1,1,1-TRIFLUORO-2-HYDROXY-3-PHENYLPROPANE DERIVATIVES F. Hoffmann-Roche AG (CH) 2010-07-14 EP disclosed
WO-2009040288-A1 1,1,1-TRIFLUORO-2-HYDROXY-3-PHENYLPROPANE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2009-04-02 WO disclosed